SCHEMBL6758586

SCHEMBL6758586

COC(=O)C(Cl)CCCC(Cl)C(=O)OC

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ZDHHC7 Q9NXF8 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
TSHR P16473 2/20 0.35
ALDH1A2 O94788 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALDH2 P05091 1/20 0.34
ALDH1A3 P47895 1/20 0.34
BIRC2 Q13490 4/20 0.33
CA14 Q9ULX7 2/20 0.33
ABCB1 P08183 1/20 0.32
KMT2A Q03164 2/20 0.31
CA12 O43570 1/20 0.31
USP2 O75604 1/20 0.31
LMNA P02545 1/20 0.31
MME P08473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2862449 0.95 ZDHHC7 (0.45) CA1CA2ZDHHC7SMN1; SMN2TSHR
SCHEMBL2862400 0.90 SMN1; SMN2 (0.42) CA1CA2ZDHHC7SMN1; SMN2TSHR
SCHEMBL7976135 0.89 CA1 (0.39) CA1CA2ZDHHC7SMN1; SMN2TSHR
SCHEMBL10733705 0.89 CA2 (0.59) CA1CA2ZDHHC7TSHRBIRC2
SCHEMBL4403214 0.87 ZDHHC7 (0.58) CA1CA2ZDHHC7BIRC2ABCB1
SCHEMBL7970891 0.87 ZDHHC7 (0.40) CA1CA2ZDHHC7SMN1; SMN2TSHR
SCHEMBL10911418 0.85 ZDHHC7 (0.61) CA1CA2ZDHHC7BIRC2ABCB1
SCHEMBL11877076 0.85 ZDHHC7 (0.43) CA1CA2ZDHHC7SMN1; SMN2TSHR
SCHEMBL11440159 0.85 ZDHHC7 (0.61) CA1CA2ZDHHC7BIRC2ABCB1
SCHEMBL11435375 0.85 ZDHHC7 (0.61) CA1CA2ZDHHC7BIRC2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210290769-A1 TAILORING SITE SPECIFICITY OF BIOCONJUGATION USING STEP-WISE ATRP ON PROTEINS CARNEGIE MELLON UNIVERSITY 2021-09-23 US claimed
WO-2020028700-A1 TAILORING SITE SPECIFICITY OF BIOCONJUGATION USING STEP-WISE ATRP ON PROTEINS RUSSELL ALAN J (US) 2020-02-06 WO claimed
US-12053529-B2 Amino-reactive positively charged ATRP initiators that maintain their positive charge during synthesis of biomacro-initiators CARNEGIE MELLON UNIVERSITY (US) 2024-08-06 US disclosed
US-20220275137-A1 TUNING PROTEIN SOLUBILITY BY POLYMER SURFACE MODIFICATION CARNEGIE MELLON UNIVERSITY 2022-09-01 US disclosed
US-20210388337-A1 PROTEIN-POLYMER CONJUGATES AND METHODS FOR THEIR PREPARATION CARNEGIE MELLON UNIVERSITY 2021-12-16 US disclosed
US-20210316001-A1 AMINO-REACTIVE POSITIVELY CHARGED ATRP INITIATORS THAT MAINTAIN THEIR POSITIVE CHARGE DURING SYNTHESIS OF BIOMACRO-INITIATORS CARNEGIE MELLON UNIVERSITY 2021-10-14 US disclosed
US-20210290769-A1 TAILORING SITE SPECIFICITY OF BIOCONJUGATION USING STEP-WISE ATRP ON PROTEINS CARNEGIE MELLON UNIVERSITY 2021-09-23 US disclosed
WO-2021022198-A1 TUNING PROTEIN SOLUBILITY BY POLYMER SURFACE MODIFICATION Carnegie Mellon University (CMU) (US) 2021-02-04 WO disclosed
WO-2020123023-A2 PROTEIN-POLYMER CONJUGATES AND METHODS FOR THEIR PREPARATION CARNEGIE MELLON UNIVERSITY (US) 2020-06-18 WO disclosed
WO-2020028715-A1 AMINO-REACTIVE POSITIVELY CHARGED ATRP INITIATORS THAT MAINTAIN THEIR POSITIVE CHARGE DURING SYNTHESIS OF BIOMACRO-INITIATORS RUSSELL ALAN J (US) 2020-02-06 WO disclosed
WO-2020028700-A1 TAILORING SITE SPECIFICITY OF BIOCONJUGATION USING STEP-WISE ATRP ON PROTEINS RUSSELL ALAN J (US) 2020-02-06 WO disclosed
US-6716918-B2 ATOM TRANSFER RADICAL POLYMERIZATION IN THE PRESENCE OF A REDOX CATALYST OF A TRANSITION METAL COMPLEX ALSO USING AN ORGANOHALOGEN OR HALOGENATED SULFONYL COMPOUND AS A POLYMERIZATION CATALYST MITSUBISHI CHEMICAL CORPORATION (JP) 2004-04-06 US disclosed
US-20040053309-A1 Proteins, genes and their use for diagnosis and treatment of kidney response OXFORD GLYCOSCIENCES (UK) LTD. (GB) 2004-03-18 US disclosed
US-20020156196-A1 Methacrylate-based polymer and process for producing the same MITSUBISHI CHEMICAL CORPORATION (JP) 2002-10-24 US disclosed