SCHEMBL6766027

SCHEMBL6766027

COc1cccc(C2=NN(c3ccccc3)C(=O)CO2)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.46
PTGS2 P35354 2/20 0.46
GAA P10253 5/20 0.43
UGCG Q16739 2/20 0.43
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
MAOB P27338 1/20 0.42
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 3/20 0.41
HSD17B10 Q99714 1/20 0.41
HIF1A Q16665 1/20 0.39
HPGD P15428 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CHRM2 P08172 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6766907 0.85 PTGS1 (0.50) PTGS1PTGS2GAAUGCGPDE4A
SCHEMBL10636445 0.80 SHMT2 (0.43) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL5778908 0.79 PTGS1 (0.46) PTGS1PTGS2GAAUGCGPDE4A
SCHEMBL10630259 0.78 GAA (0.49) PTGS1GAAALDH1A1SMN1; SMN2POLB
SCHEMBL10630291 0.76 MAOB (0.43) PTGS1GAAMAOBALDH1A1SMN1; SMN2
SCHEMBL6763490 0.76 CYP2D6 (0.54) PTGS1GAAMAOBALDH1A1SMN1; SMN2
SCHEMBL6763622 0.76 GAA (0.42) PTGS1PTGS2GAAMAOBALDH1A1
SCHEMBL10630231 0.75 PDE4A (0.52) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL10633535 0.75 APP (0.51) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL6766625 0.75 GAA (0.46) PTGS1PTGS2GAAMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825192-B1 NON-N-METHYL-D-ASPARTATE (NON- NMDA) EXCITATORY AMINO ACID RECEPTOR ANTAGONISTIC ACTION, FOR EXAMPLE 2-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) RECEPTOR ANTAGONISTIC ACTION EISAI CO., LTD. (JP) 2004-11-30 US disclosed
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP disclosed