SCHEMBL6766907

SCHEMBL6766907

COc1cccc(OC)c1C1=NN(c2ccccc2)C(=O)CO1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.50
PTGS2 P35354 3/20 0.50
GAA P10253 3/20 0.46
PDE4A P27815 3/20 0.45
PDE4B Q07343 3/20 0.45
PDE4C Q08493 3/20 0.45
PDE4D Q08499 3/20 0.45
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CHRM2 P08172 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
CHRM1 P11229 1/20 0.42
TSHR P16473 1/20 0.42
DRD3 P35462 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6766027 0.85 PTGS1 (0.46) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL5778908 0.83 PTGS1 (0.46) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL10630231 0.79 PDE4A (0.52) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL10633535 0.79 APP (0.51) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL6768350 0.77 KMT2A (0.47) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL10636445 0.76 SHMT2 (0.43) PTGS1PTGS2GAAPDE4APDE4B
SCHEMBL10633512 0.75 KMT2A (0.52) PTGS1GAAPDE4APDE4BPDE4C
SCHEMBL10630259 0.74 GAA (0.49) PTGS1GAAALDH1A1KDM4EKMT2A
SCHEMBL6763591 0.74 GAA (0.46) PTGS1GAAALDH1A1KDM4EKMT2A
SCHEMBL10633478 0.74 CES2 (0.46) PTGS1GAAALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825192-B1 NON-N-METHYL-D-ASPARTATE (NON- NMDA) EXCITATORY AMINO ACID RECEPTOR ANTAGONISTIC ACTION, FOR EXAMPLE 2-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) RECEPTOR ANTAGONISTIC ACTION EISAI CO., LTD. (JP) 2004-11-30 US disclosed
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP disclosed