SCHEMBL6770516

SCHEMBL6770516

CC(=O)Nc1ccc(S(=O)(=O)Cl)c(Br)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
CDK1 P06493 1/20 0.50
CA2 P00918 3/20 0.47
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA9 Q16790 2/20 0.47
MAPT P10636 2/20 0.46
IDO1 P14902 3/20 0.46
ATAD2 Q6PL18 1/20 0.46
CECR2 Q9BXF3 1/20 0.46
ENPP2 Q13822 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
MAOA P21397 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18239828 0.85 ALDH1A1 (0.69) ALDH1A1CDK1CA2CA12CA1
SCHEMBL539699 0.82 ALDH1A1 (0.73) ALDH1A1CDK1CA2CA12CA1
SCHEMBL686781 0.81 ALDH1A1 (0.54) ALDH1A1CDK1CA2CA12CA1
SCHEMBL1818154 0.80 CA12 (0.51) CA2CA12CA1CA9MAPT
SCHEMBL1817574 0.79 ALDH1A1 (0.53) ALDH1A1CDK1CA2CA12CA1
SCHEMBL10719928 0.79 ATAD2 (0.65) ALDH1A1CDK1MAPTIDO1ATAD2
SCHEMBL6771522 0.79 ALDH1A1 (0.59) ALDH1A1CDK1MAPTATAD2CECR2
SCHEMBL7659979 0.77 HTT (0.54) ALDH1A1CA2CA12CA1CA9
SCHEMBL20819276 0.76 CNR2 (0.54) ALDH1A1CA2CA9MAPTATAD2
SCHEMBL11481936 0.75 GAA (0.57) ALDH1A1CDK1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6673824-B1 HYPOTENSIVE AGENTS BRISTOL-MYERS SQUIBB CO. 2004-01-06 US disclosed
US-6107320-A Phenyl sulfonamide endothelin antagonists BRISTOL-MYERS SQUIBB CO. (US) 2000-08-22 US disclosed
EP-0569193-B1 N-isoxazole-phenylsulfonamide derivatives and their use as endothelin antagonists SQUIBB & SONS INC (US) 1997-02-26 EP disclosed
US-5514696-A Phenyl sulfonamide endothelin antagonists BRISTOL-MYERS SQUIBB CO. (US) 1996-05-07 US disclosed
EP-0569193-A1 N-isoxazole-phenylsulfonamide derivatives and their use as endothelin antagonists E.R. SQUIBB & SONS, INC. (US) 1993-11-10 EP disclosed