SCHEMBL6770609

SCHEMBL6770609

Fc1[c]c(Cl)c(-c2ccccc2Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.40
DPP4 P27487 1/20 0.38
HSD11B1 P28845 3/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
PTPRC P08575 1/20 0.35
LMNA P02545 2/20 0.35
TSHR P16473 1/20 0.35
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
PLA2G7 Q13093 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KCNN4 O15554 1/20 0.33
IDO1 P14902 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
PDK2 Q15119 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15637395 0.84 CYP2A6 (0.40) CYP2A6DPP4HSD11B1NPC1RAB9A
SCHEMBL10475010 0.84 PTPRC (0.34) HSD11B1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL10474986 0.82 IDO1 (0.38) HSD11B1TP53LMNAALDH1A1IDO1
SCHEMBL15637369 0.79 CYP2A6 (0.43) CYP2A6DPP4HSD11B1NPC1RAB9A
SCHEMBL11444153 0.78 NISCH (0.40) HSD11B1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL15287292 0.78 AHR (0.42) HSD11B1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL7814348 0.78 CYP2A6 (0.41) CYP2A6SMN1; SMN2HPGDLMNATSHR
SCHEMBL671133 0.72 CYP2A6 (0.67) CYP2A6DPP4HSD11B1NPC1RAB9A
SCHEMBL29883244 0.72 CYP2A6 (0.67) CYP2A6DPP4HSD11B1NPC1RAB9A
SCHEMBL29802156 0.72 CYP2A6 (0.67) CYP2A6DPP4HSD11B1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903440-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer CropScience AG (DE) 2015-08-12 EP disclosed
WO-2014053450-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2014-04-10 WO disclosed
US-6720344-B2 BINDING TO NUCLEAR RECEPTOR PROTEINS; STIMULATING BMP-2 PROMOTER ACTIVITY THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2004-04-13 US disclosed
US-20030119791-A1 Methods and compositions for stimulating osteoblast proliferation or treating malignant cell proliferation and methods for selecting osteoblast proliferation stimulants KERWIN SEAN M (US) 2003-06-26 US disclosed
EP-0912549-A4 COMPOUNDS AND METHODS FOR PROVIDING PHARMACOLOGICALLY ACTIVE PREPARATIONS AND USES THEREOF UNIV TEXAS (US) 2002-01-02 EP disclosed
EP-0912549-A1 COMPOUNDS AND METHODS FOR PROVIDING PHARMACOLOGICALLY ACTIVE PREPARATIONS AND USES THEREOF THE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1999-05-06 EP disclosed
WO-1997048694-A1 COMPOUNDS AND METHODS FOR PROVIDING PHARMACOLOGICALLY ACTIVE PREPARATIONS AND USES THEREOF BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1997-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030119791-A1 Methods and compositions for stimulating osteoblast proliferation or treating malignant cell proliferation and methods for selecting osteoblast proliferation stimulants MKI67, HGF, AREG CYP2A6 2402/4885DPP4 4106/4885HSD11B1 184/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.