SCHEMBL6772789

SCHEMBL6772789

O=S(=O)(Cl)c1cc(OCc2ccccc2)ccc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.51
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA7 P43166 2/20 0.51
CA9 Q16790 2/20 0.51
CA4 P22748 1/20 0.51
CA5A P35218 1/20 0.51
CA5B Q9Y2D0 1/20 0.51
MAOB P27338 7/20 0.50
ALOX5 P09917 1/20 0.49
MEN1 O00255 1/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 1/20 0.46
TOP1 P11387 1/20 0.46
AR P10275 4/20 0.45
MAOA P21397 5/20 0.45
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6772019 0.86 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL3823883 0.77 MAOB (0.62) CA12CA1CA2CA7CA9
SCHEMBL8665563 0.77 MAOB (0.51) CA12CA1CA2CA7CA9
SCHEMBL1461751 0.76 MAOB (0.57) MAOBALOX5MEN1KMT2ATOP1
SCHEMBL1588758 0.76 BACE1 (0.57) CA12CA1CA2CA7CA9
SCHEMBL1818122 0.75 AR (0.55) CA12CA1CA2CA7CA9
SCHEMBL1523177 0.75 CA12 (0.60) CA12CA1CA2CA7CA9
SCHEMBL2329379 0.75 ALOX5 (0.63) CA12CA1CA2CA7CA9
SCHEMBL926213 0.74 CA12 (0.70) CA12CA1CA2CA7CA9
SCHEMBL615020 0.74 MAOB (0.59) MAOBALOX5TOP1MAOARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6673824-B1 HYPOTENSIVE AGENTS BRISTOL-MYERS SQUIBB CO. 2004-01-06 US disclosed
US-6107320-A Phenyl sulfonamide endothelin antagonists BRISTOL-MYERS SQUIBB CO. (US) 2000-08-22 US disclosed
US-5514696-A Phenyl sulfonamide endothelin antagonists BRISTOL-MYERS SQUIBB CO. (US) 1996-05-07 US disclosed