SCHEMBL6773809

SCHEMBL6773809

CC#CCOc1ccc(S(=O)(=O)C(C)NC(C(=O)O)C(C)C)cc1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 19/20 0.61
MMP13 P45452 14/20 0.61
MMP9 P14780 13/20 0.61
MMP1 P03956 12/20 0.61
MMP14 P50281 2/20 0.53
ADAM10 O14672 1/20 0.53
MMP7 P09237 1/20 0.53
MMP8 P22894 1/20 0.53
MMP2 P08253 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7394268 0.90 ADAM17 (0.60) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL7396222 0.84 ADAM17 (0.54) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL6508748 0.83 MMP9 (0.79) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL6499431 0.81 ADAM17 (0.59) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL6773805 0.80 ADAM17 (0.57) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL7430744 0.80 ADAM17 (0.52) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL6265979 0.77 ADAM17 (0.60) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL3943916 0.76 ADAM17 (1.00) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL6502069 0.76 ADAM17 (0.78) ADAM17MMP13MMP9MMP1MMP14
SCHEMBL7393438 0.76 ADAM17 (0.66) ADAM17MMP13MMP9MMP1MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6812227-B2 SULFUR COMPOUNDS SUCH AS 2-((4-BUT-2-YNYLOXY-BENZENESULFONYL)-METHYL-AMINO)-N-HYDROXY-3-METHYL -BUTYRAMIDE, USED AS TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME (TACE) INHIBITORS, FOR PROPHYLAXIS OF RHEUMATIC DISEASES, SEPSIS OR INFLAMMATION WYETH HOLDINGS CORPORATION 2004-11-02 US disclosed