SCHEMBL6774198

SCHEMBL6774198

Clc1ccc(CNCCCNc2ccc3ccccc3n2)cc1Cl

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MARS1 P56192 1/20 0.49
DRD2 P14416 1/20 0.43
ADRA1A P35348 1/20 0.43
DRD3 P35462 1/20 0.43
KCNH2 Q12809 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
MC4R P32245 2/20 0.43
MC5R P33032 2/20 0.43
MC3R P41968 1/20 0.43
SSTR3 P32745 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HDAC6 Q9UBN7 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5943554 0.87 MC5R (0.57) MC4RMC5RMC3RNPC1RAB9A
SCHEMBL5943501 0.81 NPC1 (0.48) HRH4MC4RMC5RMC3RNPC1
SCHEMBL5943512 0.80 ATM (0.47) DRD2ADRA1ADRD3KCNH2HRH4
SCHEMBL27565799 0.80 MCHR1 (0.47) MARS1MC4RMC5RMC3RSSTR3
SCHEMBL10069775 0.79 DRD2 (0.44) DRD2ADRA1ADRD3KCNH2HRH4
SCHEMBL5943593 0.78 TP53 (0.42) DRD2ADRA1ADRD3KCNH2HRH4
SCHEMBL5943486 0.78 NCF1 (0.59) DRD2ADRA1ADRD3KCNH2HRH4
SCHEMBL5943562 0.78 NOS1 (0.46) NPC1RAB9AHDAC6CYP1A2CYP2D6
SCHEMBL5943504 0.78 NPC1 (0.51) DRD2ADRA1ADRD3KCNH2HRH4
SCHEMBL5943457 0.77 MCHR1 (0.53) DRD2ADRA1ADRD3KCNH2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818655-B2 2-AMINOQUINOLINES; CARDIOVASCULAR, GASTROINTESTINAL, PYSCHOLOGICAL, RESPIRATORY AND NERVOUS SYSTEM DISORDERS SMITHKLINE BEECHAM CORPORATION 2004-11-16 US disclosed