SCHEMBL6775245

SCHEMBL6775245

COc1cccc2ncc3c(c12)-c1ccncc1C3=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
SLC22A12 Q96S37 2/20 0.40
ELANE P08246 2/20 0.38
FGFR1 P11362 1/20 0.36
SRC P12931 1/20 0.36
FGFR2 P21802 1/20 0.36
FGFR4 P22455 1/20 0.36
FGFR3 P22607 1/20 0.36
CDC25B P30305 1/20 0.36
CYP19A1 P11511 3/20 0.36
GSK3B P49841 2/20 0.36
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6776178 0.75 MAOA (0.56) MAOAMAOBCYP1A2CYP3A4TSHR
SCHEMBL7265998 0.73 CCNE2 (0.41) MAOAMAOBMEN1KMT2ACYP1A2
SCHEMBL6774511 0.68 MAOA (0.46) MAOAMAOBMEN1KMT2ACYP3A4
SCHEMBL8280623 0.66 MAOA (0.61) MAOAMAOBCYP3A4TSHRELANE
SCHEMBL1649965 0.66 MAOA (0.44) MAOAMAOBMEN1KMT2ACYP3A4
SCHEMBL6775253 0.66 MAOA (0.44) MAOAMAOBMEN1KMT2ACYP1A2
SCHEMBL5780263 0.65 PDE3B (0.42) MEN1KMT2ACYP1A2CYP3A4CYP2C19
SCHEMBL20618218 0.65 MAOA (0.77) MAOAMAOBMEN1KMT2ACYP1A2
SCHEMBL8417659 0.65 MAOA (0.86) MAOAMAOBMEN1KMT2ACYP3A4
SCHEMBL31112247 0.65 MAOA (0.77) MAOAMAOBMEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6680326-B2 ANTITUMOR AGENTS; ANTICANCER AGENTS HOFFMANN-LA ROCHE INC. 2004-01-20 US disclosed