SCHEMBL6776691

SCHEMBL6776691

CC(C)COc1ncc(I)cc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.45
XDH P47989 3/20 0.41
DHODH Q02127 2/20 0.40
SLC22A12 Q96S37 1/20 0.39
NR1H4 Q96RI1 2/20 0.37
MAP3K7 O43318 1/20 0.37
TAB1 Q15750 1/20 0.37
MYC P01106 2/20 0.36
MAX P61244 2/20 0.36
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36
GCK P35557 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN9A Q15858 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6361867 0.83 KMT2A (0.49) TP53ALDH1A1TSHRKMT2A
SCHEMBL11551863 0.82 PTGER1 (0.43) TP53XDHDHODHSCN5ASCN9A
SCHEMBL2405699 0.80 TP53 (0.41) TP53DHODHALDH1A1TSHRKMT2A
SCHEMBL25704057 0.79 POLB (0.42) DHODHALDH1A1KMT2A
SCHEMBL6624693 0.79 KDM4E (0.45) TP53RARARARBRARGALDH1A1
SCHEMBL23525777 0.78 ALDH1A1 (0.46) ALDH1A1TSHR
SCHEMBL5446405 0.72 ALDH1A1 (0.49) DHODHNR1H4MYCALDH1A1TSHR
SCHEMBL7584370 0.72 XDH (0.41) TP53XDHDHODHNR1H4MAP3K7
SCHEMBL1853295 0.71 KDM4C (0.52) TP53XDHDHODHSLC22A12NR1H4
SCHEMBL7432976 0.71 ALDH1A1 (0.47) DHODHNR1H4MYCALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6756373-B1 SUCH AS 5-(2-BUTOXY-5-IODO-3-PYRIDINYL)-3-ETHYL-2-(2-METHOXY-ETHYL)-2,6-DIHYDRO-7H -PYRAZOLO(4,3-D)PYRIMIDIN-7-ONE; CYCLIC GUANOSINE 3',5'-MONOPHOSPHATE PHOSPHODIESTERASE INHIBITORS; ERECTILE DYSFUNCTION PFIZER INC. 2004-06-29 US disclosed