SCHEMBL6779241

SCHEMBL6779241

CCC(c1ccccc1)(c1ccccc1)C(O)C#N

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.45
GRIN2A Q12879 4/20 0.45
GRIN2D O15399 3/20 0.45
GRIN2C Q14957 3/20 0.45
GRIN2B Q13224 2/20 0.45
LMNA P02545 2/20 0.39
TSHR P16473 1/20 0.39
CYP2D6 P10635 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C19 P33261 1/20 0.36
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
KCNN4 O15554 1/20 0.34
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28225801 0.79 CYP2D6 (0.41) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL416118 0.78 GRIN1 (0.47) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL18251092 0.75 ALDH1A1 (0.43) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL6781624 0.75 TSHR (0.43) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL4454908 0.74 GRIN1 (0.43) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL6284917 0.71 GRIN1 (0.44) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL16428269 0.71 TSHR (0.43) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL1067596 0.70 TSHR (0.39) TSHRCYP2D6CYP3A4ALDH1A1MAPT
SCHEMBL678931 0.69 KMT2A (0.48) LMNATSHRCYP2D6CYP3A4CYP2C19
SCHEMBL14164384 0.68 GRIN1 (0.50) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6686369-B1 α-hydrdroxylic acid derivatives, their production and use ABBOTT GMBH & CO., KG (DE) 2004-02-03 US disclosed
EP-0892787-B1 NOVEL ALPHA-HYDROXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE ABBOTT GMBH & CO KG (DE) 2003-06-11 EP disclosed
EP-0892787-A1 NOVEL $g(a)-HYDROXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1999-01-27 EP disclosed
WO-1997038981-A1 NOVEL α-HYDROXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1997-10-23 WO disclosed