SCHEMBL6781256

SCHEMBL6781256

CC1=Cc2c(ccc(-c3ccccc3)c2-c2ccccc2)C1[Si](C)(C)C1C(C)=Cc2c1ccc(-c1ccccc1)c2-c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.33
BRD2 P25440 1/20 0.33
PTGS1 P23219 3/20 0.33
PTGS2 P35354 3/20 0.33
TDO2 P48775 1/20 0.32
HSP90AB1 P08238 1/20 0.31
AKT2 P31751 2/20 0.30
CHEK1 O14757 1/20 0.30
AKT1 P31749 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1453850 0.86 BRD4 (0.36) BRD4BRD2PTGS1PTGS2TDO2
SCHEMBL61908 0.84 PDCD1 (0.34) BRD4AKT2AKT1
SCHEMBL29366427 0.84 PDCD1 (0.34) BRD4AKT2AKT1
Hydrochloric Acid SCHEMBL3822639 0.82 ADRA2A (0.34) BRD4TDO2AKT2AKT1
Dimethylamine SCHEMBL1453283 0.81 TDO2 (0.33) TDO2
SCHEMBL6056122 0.78 PDCD1 (0.30)
SCHEMBL1452295 0.78 PDCD1 (0.30)
SCHEMBL16683341 0.78 PDCD1 (0.30)
SCHEMBL1452790 0.77 MAPK1 (0.39)
SCHEMBL5838399 0.77 PDK2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6730756-B1 HETEROGENEOUS TRANSITION METAL CATALYST WITH METALLOCENE IMPREGNATED BOREALIS A/S (DK) 2004-05-04 US disclosed