SCHEMBL6783499

SCHEMBL6783499

Cc1cc(CCN)c2ccccc2n1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 4/20 0.58
CYP1A2 P05177 2/20 0.56
KDM4E B2RXH2 2/20 0.48
RAB9A P51151 1/20 0.48
TAAR1 Q96RJ0 1/20 0.46
CYP2C19 P33261 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HTT P42858 2/20 0.45
BACE1 P56817 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
CYP2D6 P10635 1/20 0.44
HPGD P15428 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TLR8 Q9NR97 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14268962 0.88 TLR8 (0.54) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL265139 0.85 NCF1 (0.61) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL18535317 0.84 CYP1A2 (0.58) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL6964689 0.82 CYP1A2 (0.56) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL28728112 0.82 CYP1A2 (0.56) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL6788358 0.82 CYP2C19 (0.56) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL8232676 0.79 CYP1A2 (0.62) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL1366357 0.79 CYP1A2 (0.62) NCF1CYP1A2KDM4ERAB9ACYP2C19
SCHEMBL6788451 0.79 NCF1 (0.60) NCF1CYP1A2RAB9ATAAR1HTT
SCHEMBL6790022 0.79 NCF1 (0.60) NCF1CYP1A2KDM4ECYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825215-B2 N-HYDROXY-2-(2-(((4-((2-METHYL-4-QUINOLINYL)METHOXY)PHENYL) -SULFONYL)METHYL)-2-PYRROLIDINYL)ACETAMIDE, FOR EXAMPLE AND OTHER QUINOLINE CONTAINING N-HYDROXYACETAMIDE DERIVATIVES BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-11-30 US disclosed
EP-1355901-A2 1,1-DISUBSTITUTED CYCLIC INHIBITORS OF MATRIX METALLOPROTEASE AND TNF-$g(a) Bristol-Myers Squibb Pharma Company (US) 2003-10-29 EP disclosed
WO-2002055516-A2 1,1-DISUBSTITUTED CYCLIC INHIBITORS OF MATRIX METALLOPROTEASE AND TNF-$g(a) BRISTOL MYERS SQUIBB CO (US) 2002-07-18 WO disclosed