SCHEMBL6788451

SCHEMBL6788451

Cc1cc(CCN(C)C)c2ccccc2n1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 3/20 0.60
CYP1A2 P05177 1/20 0.53
HTT P42858 1/20 0.51
NUDT1 P36639 1/20 0.46
NPC1 O15118 2/20 0.45
SLC2A1 P11166 2/20 0.45
POLB P06746 1/20 0.45
APOBEC3A P31941 1/20 0.45
RAD52 P43351 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
APOBEC3G Q9HC16 1/20 0.45
HTR1A P08908 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
TAAR1 Q96RJ0 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6788659 0.83 CYP1A2 (0.56) NCF1CYP1A2HTTNPC1RAB9A
SCHEMBL18535317 0.81 CYP1A2 (0.58) NCF1CYP1A2HTTRAB9A
SCHEMBL6783499 0.79 NCF1 (0.58) NCF1CYP1A2HTTPOLBRAB9A
SCHEMBL6964689 0.79 CYP1A2 (0.56) NCF1CYP1A2HTTRAB9AKMT2A
SCHEMBL6788358 0.79 CYP2C19 (0.56) NCF1CYP1A2HTTRAB9AKMT2A
SCHEMBL28728112 0.79 CYP1A2 (0.56) NCF1CYP1A2HTTRAB9AKMT2A
SCHEMBL14408133 0.78 NCF1 (0.48) NCF1CYP1A2HTTNPC1SLC2A1
SCHEMBL1366357 0.77 CYP1A2 (0.62) NCF1CYP1A2HTTRAB9AKMT2A
SCHEMBL8232676 0.77 CYP1A2 (0.62) NCF1CYP1A2HTTRAB9AKMT2A
SCHEMBL6789734 0.77 CYP1A2 (0.53) NCF1CYP1A2HTTRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825215-B2 N-HYDROXY-2-(2-(((4-((2-METHYL-4-QUINOLINYL)METHOXY)PHENYL) -SULFONYL)METHYL)-2-PYRROLIDINYL)ACETAMIDE, FOR EXAMPLE AND OTHER QUINOLINE CONTAINING N-HYDROXYACETAMIDE DERIVATIVES BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-11-30 US disclosed
EP-1355901-A2 1,1-DISUBSTITUTED CYCLIC INHIBITORS OF MATRIX METALLOPROTEASE AND TNF-$g(a) Bristol-Myers Squibb Pharma Company (US) 2003-10-29 EP disclosed
WO-2002055516-A2 1,1-DISUBSTITUTED CYCLIC INHIBITORS OF MATRIX METALLOPROTEASE AND TNF-$g(a) BRISTOL MYERS SQUIBB CO (US) 2002-07-18 WO disclosed