SCHEMBL678490

SCHEMBL678490

Cn1nc(-c2cccnc2)cc1-c1cccc(-c2ncccn2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 8/20 0.46
CYP2E1 P05181 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2B6 P20813 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP19A1 P11511 2/20 0.43
GRM5 P41594 1/20 0.43
FYN P06241 2/20 0.41
CYP3A4 P08684 3/20 0.41
USP8 P40818 1/20 0.41
KARS1 Q15046 1/20 0.40
HTR2C P28335 1/20 0.40
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2731043 0.90 CYP2A6 (0.44) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12278093 0.88 CYP2A6 (0.48) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12278716 0.86 CYP2A6 (0.51) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12279610 0.83 USP8 (0.47) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12279439 0.80 CYP2A6 (0.54) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL13989135 0.80 CYP2A6 (0.62) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12278130 0.76 CYP2A6 (0.45) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL28049612 0.76 CYP2A6 (0.57) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12279662 0.75 CYP2A6 (0.47) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12278719 0.75 CYP2A6 (0.42) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9451775-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-09-27 US disclosed
US-9451775-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-09-27 US disclosed
EP-2586312-B1 Heterocyclic compounds as pest controllers BAYER CROPSCIENCE AG (DE) 2016-04-27 EP disclosed
US-20140336186-A1 Heterocyclic Compounds as Pesticides BAYER CORPSCIENCE AG (DE) 2014-11-13 US disclosed
US-20140336186-A1 Heterocyclic Compounds as Pesticides BAYER CORPSCIENCE AG (DE) 2014-11-13 US disclosed
US-8809547-B2 Heterocyclic compounds as pesticides BAYER CROPSCIENCE AG (DE) 2014-08-19 US disclosed
US-8809547-B2 Heterocyclic compounds as pesticides BAYER CROPSCIENCE AG (DE) 2014-08-19 US disclosed
EP-2591674-A1 Heterocyclic compounds as pest controllers Bayer CropScience AG (DE) 2013-05-15 EP disclosed
EP-2586311-A1 Heterocyclic compounds as pest controllers Bayer CropScience AG (DE) 2013-05-01 EP disclosed
EP-2586312-A1 Heterocyclic compounds as pest controllers Bayer CropScience AG (DE) 2013-05-01 EP disclosed
EP-2583556-A1 Heterocyclic compounds as pest controllers Bayer CropScience AG (DE) 2013-04-24 EP disclosed
EP-2583557-A1 Heterocyclic compounds as pest controllers Bayer CropScience AG (DE) 2013-04-24 EP disclosed
US-20110275583-A1 Synergistic active compound combinations BAYER CROPSCIENCE AG (DE) 2011-11-10 US disclosed
US-20110275583-A1 Synergistic active compound combinations BAYER CROPSCIENCE AG (DE) 2011-11-10 US disclosed
WO-2011134964-A1 SYNERGISTIC ACTIVE SUBSTANCE COMBINATIONS BAYER CROPSCIENCE AG (DE) 2011-11-03 WO disclosed
EP-2382865-A1 Synergistic active agent compounds Bayer CropScience AG (DE) 2011-11-02 EP disclosed
US-20110212949-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG 2011-09-01 US disclosed
US-20110212949-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG 2011-09-01 US disclosed
WO-2010006713-A2 HETEROCYCLIC COMPOUNDS USED AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2010-01-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212949-A1 Heterocyclic Compounds as Pesticides DDT, ACHE, PTMS CYP2A6 277/4885CYP2E1 26/4885CYP2C9 49/4885
US-20140336186-A1 Heterocyclic Compounds as Pesticides DDT, ACHE, PTMS CYP2A6 277/4885CYP2E1 26/4885CYP2C9 49/4885
US-20110275583-A1 Synergistic active compound combinations ACHE, ACAT2, ACAT1 CYP2A6 794/4885CYP2E1 531/4885CYP2C9 827/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.