SCHEMBL6786929

SCHEMBL6786929

Cc1cc(C)n2c(cc3ccccc32)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.44
NPC1 O15118 5/20 0.44
RAB9A P51151 5/20 0.44
SMN1; SMN2 Q16637 4/20 0.43
PBRM1 Q86U86 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GAA P10253 2/20 0.41
MAPT P10636 4/20 0.41
PIK3CG P48736 1/20 0.41
ALDH1A1 P00352 6/20 0.40
HPGD P15428 4/20 0.40
SLC6A2 P23975 1/20 0.38
POLB P06746 1/20 0.37
TSHR P16473 3/20 0.37
HSD17B10 Q99714 2/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19787889 0.80 MAPT (0.53) KDM4ENPC1RAB9ASMN1; SMN2PBRM1
SCHEMBL29449194 0.73 KDM4E (0.57) KDM4ENPC1RAB9ASMN1; SMN2GAA
SCHEMBL11628053 0.70 SMN1; SMN2 (0.51) KDM4ENPC1RAB9ASMN1; SMN2PBRM1
SCHEMBL29511771 0.67 SMN1; SMN2 (0.41) KDM4ESMN1; SMN2PBRM1L3MBTL1ALDH1A1
SCHEMBL29354440 0.67 SMN1; SMN2 (0.39) KDM4ESMN1; SMN2PBRM1L3MBTL1MAPT
SCHEMBL4510784 0.67 SMN1; SMN2 (0.39) KDM4ESMN1; SMN2PBRM1L3MBTL1MAPT
SCHEMBL1772021 0.67 SMN1; SMN2 (0.61) KDM4ERAB9ASMN1; SMN2PBRM1L3MBTL1
SCHEMBL19787891 0.66 SMN1; SMN2 (0.39) KDM4ENPC1SMN1; SMN2PBRM1L3MBTL1
SCHEMBL30649148 0.66 TERT (0.36) KDM4ESMN1; SMN2PBRM1L3MBTL1GAA
SCHEMBL13852989 0.64 KMT2A (0.41) KDM4ESMN1; SMN2PBRM1L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999065902-A1 METHOD FOR PRODUCING 2,4-DIMETHYLCARBOLINE AND 2,4-DIMETHYLPYRIMIDO[1,2-a]INDOLE BAYER AKTIENGESELLSCHAFT (DE) 1999-12-23 WO claimed
US-6774236-B1 METHYLBENZENEACETIC ACID ESTER DERIVATIVES AS CHEMICAL INTERMEDIATES BAYER AKTIENGESELLSCHAFT (DE) 2004-08-10 US disclosed
EP-0799829-B1 Process for the preparation of enantiomerically pure cycloalkanoindole-, azaindole- and pyrimido [1,2a] indole carboxylic acids and their activated derivatives BAYER AG (DE) 2003-07-30 EP disclosed
WO-1999065902-A1 METHOD FOR PRODUCING 2,4-DIMETHYLCARBOLINE AND 2,4-DIMETHYLPYRIMIDO[1,2-a]INDOLE BAYER AKTIENGESELLSCHAFT (DE) 1999-12-23 WO disclosed
WO-1999065902-A1 METHOD FOR PRODUCING 2,4-DIMETHYLCARBOLINE AND 2,4-DIMETHYLPYRIMIDO[1,2-a]INDOLE BAYER AKTIENGESELLSCHAFT (DE) 1999-12-23 WO disclosed
WO-1999065902-A1 METHOD FOR PRODUCING 2,4-DIMETHYLCARBOLINE AND 2,4-DIMETHYLPYRIMIDO[1,2-a]INDOLE BAYER AKTIENGESELLSCHAFT (DE) 1999-12-23 WO disclosed
US-5952498-A SYNTHESIZING THE CHEMICAL INTERMEDIATES FOR ANTIATHEROSCLEROTICALLY ACTIVE DRUG BAYER AKTIENGESELLSCHAFT (DE) 1999-09-14 US disclosed
EP-0799829-A1 Process for the preparation of enantiomerically pure cycloalkanoindole-, azaindole- and pyrimido [1,2a] indole carboxylic acids and their activated derivatives BAYER AG (DE) 1997-10-08 EP disclosed