SCHEMBL67880

SCHEMBL67880

CCOC(=O)C1(c2ccccc2)CCCC1OCCN(CC)CC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRCP P42785 2/20 0.54
SIGMAR1 Q99720 2/20 0.54
ALDH1A1 P00352 5/20 0.53
POLB P06746 1/20 0.53
CHRM2 P08172 7/20 0.50
CHRM1 P11229 6/20 0.50
CYP3A4 P08684 4/20 0.50
LMNA P02545 3/20 0.50
CYP1A2 P05177 3/20 0.50
CYP2D6 P10635 3/20 0.50
TSHR P16473 3/20 0.50
SLC22A1 O15245 2/20 0.50
KDM4E B2RXH2 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
THRB P10828 1/20 0.50
HTT P42858 1/20 0.50
TMEM97 Q5BJF2 1/20 0.50
OPRM1 P35372 3/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27655505 0.82 ADAM17 (0.48) CYP3A4CYP2D6SLC22A1KDM4EOPRM1
SCHEMBL4813929 0.79 SLC22A1 (0.50) SLC22A1OPRM1ADRA1AKCNH2OPRD1
SCHEMBL29204727 0.78 SLC22A1 (0.54) PRCPSIGMAR1SLC22A1OPRM1ADRA1A
SCHEMBL27634423 0.77 ADAM17 (0.48) CYP3A4LMNACYP2D6SLC22A1KDM4E
SCHEMBL4808702 0.75 SLC22A1 (0.46) SLC22A1OPRM1ADRA1AKCNH2OPRD1
SCHEMBL4813759 0.75 SLC22A1 (0.46) CYP3A4LMNACYP1A2CYP2D6SLC22A1
SCHEMBL8320731 0.73 SLC22A1 (0.51) SLC22A1OPRM1ADRA1AKCNH2OPRD1
SCHEMBL7164271 0.72 CHRM2 (0.54) PRCPSIGMAR1ALDH1A1POLBCHRM2
SCHEMBL4815215 0.72 SLC22A1 (0.43) LMNASLC22A1TDP1OPRM1OPRD1
SCHEMBL4810643 0.72 SLC22A1 (0.43) SLC22A1KDM4EOPRM1ADRA1AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4774 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-12296043-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2025-05-13 US claimed
EP-4510999-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS Bristol-Myers Squibb Company (US) 2025-02-26 EP claimed
US-20240165020-A1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2024-05-23 US claimed
EP-4360653-A2 LIQUISOFT CAPSULES Patheon Softgels Inc. (US) 2024-05-01 EP claimed
US-11872307-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2024-01-16 US claimed
EP-3682872-B1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2024-01-03 EP claimed
WO-2023205619-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-10-26 WO claimed
US-20220211616-A1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2022-07-07 US claimed
EP-1931320-B1 MICROPARTICLES WITH MODIFIED RELEASE OF AT LEAST ONE ACTIVE PRINCIPLE AND ORAL DOSAGE FORM COMPRISING THE SAME FLAMEL IRELAND LTD (IE) 2022-06-15 EP claimed
EP-0371085-A1 DEXTROMETHORPHAN POTENTIATOR FOR ANTICONVULSANT COMPOSITION AND METHOD PONTECORVO, Michael (US) 1990-06-06 EP claimed
EP-0219458-B1 MEDICAMENT ADSORBATES AND THEIR PREPARATION WARNER-LAMBERT COMPANY (US) 1990-05-23 EP claimed
US-4906638-A Dextromethorphan potentiator for anticonvulsant composition and method NOVA PHARMACEUTICAL CORPORATION (US) 1990-03-06 US claimed
WO-1989005641-A1 DEXTROMETHORPHAN POTENTIATOR FOR ANTICONVULSANT COMPOSITION AND METHOD PONTECORVO MICHAEL J (US) 1989-06-29 WO claimed
EP-0132472-B1 MEDICATED PRODUCTS CONTAINING A MAGNESIUM TRISILICATE ADSORBENT WITH A MEDICAMENT DRUG ADSORBED THEREON WARNER-LAMBERT COMPANY (US) 1989-06-21 EP claimed
EP-0233932-A4 ANTICONVULSANT COMPOSITIONS AND METHOD. UNIV NEW YORK (US) 1988-04-26 EP claimed
US-4694010-A DIPHENYLHYDANTOIN AS POTENTIATOR FOR DEXTROMETHORPHAN AS ANTIEPILEPTIC NEW YORK UNIVERSITY (US) 1987-09-15 US claimed
EP-0233932-A1 ANTICONVULSANT COMPOSITIONS AND METHOD NEW YORK UNIVERSITY (US) 1987-09-02 EP claimed
WO-1987001036-A1 ANTICONVULSANT COMPOSITIONS AND METHOD NEW YORK UNIVERSITY (US) 1987-02-26 WO claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed