Ladostigil

Ladostigil

SCHEMBL678895

C#CCN[C@@H]1CCc2ccc(OC(=O)N(C)CC)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACHE P22303 19/20 1.00
MAOA P21397 2/20 1.00
MAOB P27338 2/20 1.00
BCHE P06276 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ladostigil SCHEMBL3301711 1.00 ACHE (1.00) ACHEMAOAMAOBBCHE
Ladostigil SCHEMBL3893996 1.00 ACHE (1.00) ACHEMAOAMAOBBCHE
SCHEMBL13853627 0.94 ACHE (1.00) ACHEMAOAMAOBBCHE
Ladostigil SCHEMBL2387320 0.93 ACHE (0.87) ACHEMAOAMAOBBCHE
Ladostigil SCHEMBL30579760 0.93 ACHE (0.87) ACHEMAOAMAOBBCHE
SCHEMBL12043626 0.92 ACHE (0.84) ACHEMAOAMAOBBCHE
SCHEMBL13853626 0.92 ACHE (0.84) ACHEMAOAMAOBBCHE
SCHEMBL3895981 0.90 ACHE (0.98) ACHEMAOAMAOBBCHE
SCHEMBL3895985 0.90 ACHE (0.98) ACHEMAOAMAOBBCHE
SCHEMBL13449663 0.90 ACHE (0.98) ACHEMAOAMAOBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 544 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4719474-A1 METHOD OF TREATING FIBROTIC-RELATED CONDITION Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2026-04-08 EP claimed
US-12594388-B2 Device to deliver a predetermined amount of a substance to a natural orifice of the body APTARGROUP, INC. (US) 2026-04-07 US claimed
US-20250235641-A1 DEVICE TO DELIVER A PREDETERMINED AMOUNT OF A SUBSTANCE TO A NATURAL ORIFICE OF THE BODY APTARGROUP INC. (US) 2025-07-24 US claimed
US-20250205239-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING NEURODEGENERATIVE DISEASES ARIBIO CO LTD (KR) 2025-06-26 US claimed
WO-2025134070-A1 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISORDERS ARIBIO CO., LTD. (KR) 2025-06-26 WO claimed
US-20250186415-A1 EXTENDED-RELEASE PHARMACEUTICAL COMPOSITIONS FOR TREATING EYE CONDITIONS FIFTH THIRD BANK, NATIONAL ASSOCIATION, AS AGENT 2025-06-12 US claimed
US-20250152547-A1 COMPOSITIONS FOR DELIVERY OF LADOSTIGIL YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2025-05-15 US claimed
EP-4543454-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING NEURODEGENERATIVE DISEASES Aribio Co., Ltd (KR) 2025-04-30 EP claimed
CN-119524129-A Monoamine oxidase inhibitors as modulators of beta cell vulnerability in type 1 diabetes 乔斯林糖尿病中心 2025-02-28 CN claimed
US-20250032503-A1 USE OF APREPITANT FOR TREATING ALZHEIMER'S DISEASE HOTH THERAPEUTICS, INC. 2025-01-30 US claimed
WO-2022164694-A1 FIXED DOSE COMBINATION OF CHOLINESTERASE INHIBITOR AND A QUATERNARY AMMONIUM ANTIMUSCARINIC AGENT TO TREAT NEURODEGENERATIVE COGNITIVE DISORDERS QAAM PHARMACEUTICALS, LLC (US) 2022-08-04 WO claimed
US-20220226276-A1 COMPOSITIONS FOR DELIVERY OF LADOSTIGIL YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2022-07-21 US claimed
US-11383048-B2 Device to deliver a predetermined amount of a substance to a natural orifice of the body SIPNOSE LTD. (IL) 2022-07-12 US claimed
US-20220175818-A1 Inhibition of Monoamine Oxidase Subtype A (MAOA) Mitigates Cardiovascular Calcification THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2022-06-09 US claimed
EP-3980005-A1 CARABACHOL-BROMONIDINE FORMULATION TO ENHANCE ANTI-PRESBYOPIA EFFECTS Visus Therapeutics, Inc. (US) 2022-04-13 EP claimed
US-20220107305-A1 Companion Diagnostics for NSAIDS and Donepezil for Treating Specific Subpopulations of Patients Suffering from Alzheimer's Disease UNIVERSITY OF NORTH TEXAS HEALTH SCIENCE CENTER AT FORT WORTH 2022-04-07 US claimed
EP-3976188-A1 COMPOSITIONS FOR DELIVERY OF LADOSTIGIL Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2022-04-06 EP claimed
EP-3965732-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATING PRESBYOPIA AND METHODS FOR FABRICATING THEREOF Harrow IP, LLC (US) 2022-03-16 EP claimed
CN-113993584-A Compositions for delivering ladostigil 耶路撒冷希伯来大学伊森姆研究发展有限公司 2022-01-28 CN claimed
EP-1956904-B1 LOW-DOSE LADOSTIGIL FOR THE TREATMENT OF MILD COGNITIVE IMPAIRMENT YISSUM RES DEV CO (IL) 2017-04-12 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12594388-B2 Device to deliver a predetermined amount of a substance to a natural orifice of the body TNF, PYCARD, VAPA ACHE 4349/4885MAOA 4117/4885MAOB 4475/4885
US-20250032503-A1 USE OF APREPITANT FOR TREATING ALZHEIMER'S DISEASE TACR1, ACHE, TACR2 ACHE 2/4885MAOA 624/4885MAOB 755/4885
US-20220226276-A1 COMPOSITIONS FOR DELIVERY OF LADOSTIGIL DDOST, AREG, FABP2 ACHE 977/4885MAOA 3631/4885MAOB 3685/4885
US-20250152547-A1 COMPOSITIONS FOR DELIVERY OF LADOSTIGIL DDOST, AREG, FABP2 ACHE 977/4885MAOA 3631/4885MAOB 3685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.