SCHEMBL6790604

SCHEMBL6790604

COc1cccc2c1C=C(C(=O)O)C(C(F)C(F)F)O2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
NR1H4 Q96RI1 1/20 0.35
PTGS2 P35354 11/20 0.34
PTGS1 P23219 10/20 0.34
NR3C1 P04150 2/20 0.33
EDNRA P25101 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
AR P10275 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6094173 0.78 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL6092923 0.78 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL6790598 0.75 PTGS2 (0.38) CA12CA1CA2CA7CA9
SCHEMBL6790596 0.74 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL5648251 0.71 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL5644179 0.68 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL5644840 0.66 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL7145945 0.66 PTGS2 (0.41) CA12CA1CA2CA7CA9
SCHEMBL19400217 0.65 AR (0.40) CA12CA1CA2CA7CA9
SCHEMBL5763911 0.64 NR1H4 (0.62) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6806288-B1 CYCLOOXYGENASE-2 MEDIATED DISORDERS; REDUCES INFLAMMATION; FEWER SIDE EFFECTS G.D. SEARLE & CO. 2004-10-19 US disclosed