SCHEMBL6796795

SCHEMBL6796795

O=C(NC(CO)Cc1ccccc1)c1cccnc1NS(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.45
ROCK2 O75116 2/20 0.45
RPS6KA5 O75582 2/20 0.45
RPS6KA4 O75676 2/20 0.45
PRKACA P17612 2/20 0.45
MAPK1 P28482 2/20 0.45
GSK3B P49841 2/20 0.45
PRKX P51817 2/20 0.45
ROCK1 Q13464 2/20 0.45
PRKG1 Q13976 2/20 0.45
CLK4 Q9HAZ1 2/20 0.45
LIMK1 P53667 1/20 0.45
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
TDP1 Q9NUW8 2/20 0.44
GLO1 Q04760 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6796785 1.00 PDE10A (0.45) PDE10AROCK2RPS6KA5RPS6KA4PRKACA
SCHEMBL7786988 0.86 BCL2 (0.51) MEN1KMT2AKEAP1NFE2L2F2
SCHEMBL7786990 0.86 BCL2 (0.51) MEN1KMT2AKEAP1NFE2L2F2
SCHEMBL6799602 0.86 CAPN1 (0.56) MEN1KMT2ATDP1GLO1KEAP1
SCHEMBL6799603 0.86 CAPN1 (0.56) MEN1KMT2ATDP1GLO1KEAP1
SCHEMBL7789330 0.80 ALDH1A1 (0.57) ROCK2RPS6KA5RPS6KA4PRKACAMAPK1
SCHEMBL7789327 0.80 ALDH1A1 (0.57) ROCK2RPS6KA5RPS6KA4PRKACAMAPK1
SCHEMBL7787038 0.80 PKM (0.54) MEN1KMT2ASMN1; SMN2HTTF2
SCHEMBL7789864 0.80 MEN1 (0.52) MEN1KMT2ASMN1; SMN2F2PIN1
SCHEMBL7789865 0.80 MEN1 (0.52) MEN1KMT2ASMN1; SMN2F2PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040097508-A1 Novel heterocyclically substituted amides, their preparation and use ABBOTT GMBH & CO. KG (DE) 2004-05-20 US disclosed
US-6630493-B1 Inhibitors of capain enzymes useful for the treatment of ischemias of the heart, the kidney or of central nervous system (e.g. \"stroke\"), inflammations, muscular dystrophy, cataracts of the eyes, Alzheimer's disease etc. BASF AKTIENGESELLSCHAFT (DE) 2003-10-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040097508-A1 Novel heterocyclically substituted amides, their preparation and use CAPN1, CAPNS1, CAPN2 PDE10A 2667/4885ROCK2 3278/4885RPS6KA5 670/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.