SCHEMBL680159

SCHEMBL680159

CS(=O)(=O)NC(=O)c1ccc(Oc2ccccc2F)cc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 1/20 0.59
PARP10 Q53GL7 1/20 0.58
BCL2L1 Q07817 2/20 0.50
MCL1 Q07820 2/20 0.50
SCN9A Q15858 4/20 0.47
LPAR1 Q92633 7/20 0.46
LPAR5 Q9H1C0 7/20 0.46
SCN3A Q9NY46 1/20 0.46
SCN2B O60939 1/20 0.46
SCN1B Q07699 1/20 0.46
SCN5A Q14524 1/20 0.46
PTPN1 P18031 1/20 0.45
MMP1 P03956 1/20 0.45
MMP13 P45452 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681087 0.89 SCN9A (0.54) CXCL8PARP10BCL2L1MCL1SCN9A
SCHEMBL679902 0.86 SCN9A (0.56) CXCL8PARP10BCL2L1MCL1SCN9A
SCHEMBL679956 0.84 MAPK14 (0.55) BCL2L1MCL1SCN9ALPAR1LPAR5
SCHEMBL679939 0.84 MEN1 (0.60) BCL2L1MCL1SCN9ALPAR1LPAR5
SCHEMBL703171 0.84 BCL2L1 (0.59) BCL2L1MCL1SCN9ASCN3ASCN2B
SCHEMBL680618 0.83 MAPK14 (0.54) SCN9ALPAR1LPAR5SCN3A
SCHEMBL680642 0.83 SCN9A (0.50) SCN9ASCN5APTPN1MMP13
SCHEMBL679137 0.83 RORC (0.52) BCL2L1MCL1SCN9ASCN3ASCN5A
SCHEMBL680339 0.81 KMT2A (0.51) BCL2L1MCL1SCN9ASCN3APTPN1
SCHEMBL680203 0.81 SCN3A (0.45) BCL2L1MCL1SCN9ASCN3APTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010207-A1 Chemical Compounds SCN1A, SCN1B, SCN7A CXCL8 3732/4885PARP10 1389/4885BCL2L1 3284/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.