SCHEMBL6801736

SCHEMBL6801736

N#Cc1ccc(N(C(=O)c2ccc(OS(N)(=O)=O)cc2)c2ccc(OS(N)(=O)=O)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.65
CA2 P00918 2/20 0.65
CA9 Q16790 2/20 0.65
CA12 O43570 1/20 0.58
CYP19A1 P11511 11/20 0.50
STS P08842 8/20 0.50
PARP15 Q460N3 1/20 0.46
PARP10 Q53GL7 1/20 0.46
PARP2 Q9UGN5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6799997 0.89 STS (0.62) CA1CA2CA9CA12STS
SCHEMBL6799571 0.87 CA1 (0.61) CA1CA2CA9CA12CYP19A1
SCHEMBL2233585 0.86 CA2 (0.69) CA1CA2CA9CA12CYP19A1
SCHEMBL6795598 0.83 MEN1 (0.60) CA1CA2CA9CA12CYP19A1
SCHEMBL6799562 0.82 CYP19A1 (0.63) CA1CA2CA9CYP19A1STS
SCHEMBL6802989 0.81 STS (0.64) CA1CA2CA9CA12STS
SCHEMBL9451286 0.81 CA2 (1.00) CA1CA2CA9CA12CYP19A1
SCHEMBL6799672 0.79 NSD2 (0.64) CA1CA2CA9CA12CYP19A1
SCHEMBL6800721 0.78 MEN1 (0.63) CA1CA2CA9CA12CYP19A1
SCHEMBL2112966 0.76 CA2 (0.55) CA1CA2CA9CA12CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6762205-B1 STEROID SULFATASE INHIBITORS WITHOUT ESTROGENIC SIDE EFFECT ACTION TEIKOKU HORMONE MFG. CO., LTD. (JP) 2004-07-13 US disclosed
EP-1193250-A1 PHENYL SULFAMATE DERIVATIVES Teikoku Hormone Mfg. Co., Ltd. (JP) 2002-04-03 EP disclosed