SCHEMBL6799571

SCHEMBL6799571

CN(C(=O)c1ccc(OS(N)(=O)=O)cc1)c1ccc(C#N)cc1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.61
CA2 P00918 4/20 0.61
CA9 Q16790 4/20 0.61
CA12 O43570 3/20 0.59
CYP19A1 P11511 10/20 0.49
STS P08842 7/20 0.49
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46
PGR P06401 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802010 0.89 STS (0.60) CA1CA2CA9CA12STS
SCHEMBL6801736 0.87 CA1 (0.65) CA1CA2CA9CA12CYP19A1
SCHEMBL6800382 0.82 MCHR1 (0.55) HSD17B1HSD17B2PGR
SCHEMBL6799672 0.81 NSD2 (0.64) CA1CA2CA9CA12CYP19A1
SCHEMBL6795598 0.81 MEN1 (0.60) CA1CA2CA9CA12CYP19A1
SCHEMBL6799562 0.80 CYP19A1 (0.63) CA1CA2CA9CYP19A1STS
SCHEMBL2233585 0.79 CA2 (0.69) CA1CA2CA9CA12CYP19A1
SCHEMBL9451286 0.78 CA2 (1.00) CA1CA2CA9CA12CYP19A1
SCHEMBL6794239 0.78 CA2 (0.52) CA1CA2CA9CA12PGR
Water SCHEMBL11222637 0.76 PGR (0.50) CA1CA2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6762205-B1 STEROID SULFATASE INHIBITORS WITHOUT ESTROGENIC SIDE EFFECT ACTION TEIKOKU HORMONE MFG. CO., LTD. (JP) 2004-07-13 US disclosed
EP-1193250-A1 PHENYL SULFAMATE DERIVATIVES Teikoku Hormone Mfg. Co., Ltd. (JP) 2002-04-03 EP disclosed