SCHEMBL6802001

SCHEMBL6802001

NC(=O)COc1cnc2ccccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.50
ACACA Q13085 1/20 0.50
KDM4E B2RXH2 2/20 0.49
KMT2A Q03164 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MGAM O43451 1/20 0.49
PDK2 Q15119 1/20 0.48
PTPN7 P35236 1/20 0.45
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
NOTUM Q6P988 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNA4 P43681 1/20 0.44
LMNA P02545 2/20 0.44
PKM P14618 1/20 0.44
CFTR P13569 1/20 0.43
PDE10A Q9Y233 1/20 0.42
KDR P35968 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14273081 0.86 PTPN7 (0.63) RAB9AACACAKDM4EKMT2ASMN1; SMN2
SCHEMBL5266847 0.81 MGAM (0.51) RAB9AKDM4EKMT2ASMN1; SMN2MGAM
SCHEMBL159056 0.80 ALDH1A1 (0.56) RAB9AACACAKDM4EKMT2ASMN1; SMN2
SCHEMBL1478177 0.78 PTPN7 (0.71) RAB9AKMT2APTPN7NPSR1LMNA
SCHEMBL30439679 0.78 PTPN7 (0.71) RAB9AKMT2APTPN7NPSR1LMNA
SCHEMBL2345799 0.76 MGAM (0.57) RAB9AKDM4EKMT2ASMN1; SMN2MGAM
SCHEMBL13302131 0.75 RAB9A (0.55) RAB9AKDM4EKMT2ASMN1; SMN2MGAM
SCHEMBL272613 0.75 PDGFRB (0.51) RAB9AKDM4EKMT2ASMN1; SMN2MGAM
SCHEMBL28286268 0.75 PDGFRB (0.51) RAB9AKDM4EKMT2ASMN1; SMN2MGAM
SCHEMBL28028944 0.75 PDGFRB (0.51) RAB9AKDM4EKMT2ASMN1; SMN2MGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6743794-B2 MULTIDRUG RESISTANCE PROTEIN; CANCER; 3-(9-CHLORO-3-METHYL-4-OXO-5H-ISOXAZOLO(4,3-C)QUINOLIN-5-YL)) CYCLOHEXYL)-2-PIPERIDYLACETAMIDE ELI LILLY AND COMPANY 2004-06-01 US disclosed