Lisofylline

Lisofylline

SCHEMBL680306

CC(O)CCCCn1c(=O)c2c(ncn2C)n(C)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 7/20 0.67
TNF P01375 4/20 0.67
USP2 O75604 1/20 0.67
LMNA P02545 1/20 0.67
CYP1A2 P05177 1/20 0.67
TSHR P16473 1/20 0.67
NFKB1 P19838 1/20 0.67
ACHE P22303 1/20 0.67
PDE4A P27815 1/20 0.67
PMP22 Q01453 1/20 0.67
PDE4B Q07343 1/20 0.67
PDE4C Q08493 1/20 0.67
PDE4D Q08499 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
RXFP1 Q9HBX9 1/20 0.67
CHIT1 Q13231 1/20 0.58
CHIA Q9BZP6 1/20 0.58
AKR1B1 P15121 1/20 0.56
GLA P06280 1/20 0.55
BLM P54132 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lisofylline, (S)- SCHEMBL1495100 1.00 ADORA2B (0.67) ADORA2BTNFUSP2LMNACYP1A2
Lisofylline SCHEMBL39131 1.00 ADORA2B (0.67) ADORA2BTNFUSP2LMNACYP1A2
SCHEMBL6778207 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2
SCHEMBL6778919 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2
SCHEMBL6777369 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2
SCHEMBL8699282 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2
SCHEMBL6783783 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2
SCHEMBL8700060 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2
SCHEMBL6774460 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2
Lisofylline SCHEMBL10517408 0.99 ADORA2B (0.66) ADORA2BTNFUSP2LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1759 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
US-11345956-B2 Methods and compositions related to prostate cancer therapeutics THE JOHNS HOPKINS UNIVERSITY (US) 2022-05-31 US claimed
US-6710051-B1 SUBSTANCES IS A XANTHINE AND IS ADMINISTERED IN A DOSAGE OF 7.5-750 MG 1-4 TIMES DAILY TO TREAT MYOPIA KLAUS TRIER APS (DK) 2004-03-23 US claimed
US-20040013609-A1 For identification of substances for treatment or prevention of insufficient longitudinal growth of eye(hypermetropia) or excessive longitudinal growth of eye(myopia); involves measurement of effect on retinal pigment epithelium TRIER KLAUS (DK) 2004-01-22 US claimed
EP-0584347-B1 ENANTIOMERIC HYDROXYLATED XANTHINE COMPOUNDS CELL THERAPEUTICS INC (US) 2003-01-15 EP claimed
US-6294350-B1 TREATING DISEASE CHARACTERIZED BY INCREASED LEVELS OF C-JUN HOMODIMERS, INCREASED HETERODIMERIZATION OF C-JUN WITH ANOTHER SIGNALING PEPTIDE, INCREASED LEVELS OF PHOSPHORYLATED C-JUN, AND/OR INCREASED PRESENCE OF JUN KINASE DALHOUSIE UNIVERSITY (CA) 2001-09-25 US claimed
WO-2001032156-A2 METHODS FOR TREATING FIBROPROLIFERATIVE DISEASES DALHOUSIE UNIVERSITY (CA) 2001-05-10 WO claimed
WO-2000066101-A2 METHOD OF INHIBITING GLYCATION PRODUCT FORMATION CITY OF HOPE (US) 2000-11-09 WO claimed
US-5112827-A Purine derivatives, pentoxifylline, anticholesterol, arterial antideposit agents BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1992-05-12 US claimed
EP-0462506-A1 Pharmaceutical preparations of mixtures comprising cefotaxim and derivatives of xanthine and their use Schrinner, Elmar J., Dr. (DE) 1991-12-27 EP claimed
EP-0169466-B1 MIXTURE OF XANTHIN DERIVATIVES AND O-ACETYL-SALICYLIC ACID, OR THEIR PHARMACOLOGICALLY ACCEPTABLE SALTS, AND ITS USE HOECHST AKTIENGESELLSCHAFT (DE) 1990-04-04 EP claimed
US-4880791-A BLOOD DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1989-11-14 US claimed
EP-0305743-A2 Pharmaceutical mixture preparation, its manufacture and use HOECHST AKTIENGESELLSCHAFT (DE) 1989-03-08 EP claimed
US-4636507-A Host defense mechanism enhancement HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-01-13 US claimed
US-4576947-A HYDROXYALKYLXANTHINES, INCREASING CEREBRAL BLOOD FLOW, BRONCHODILATORS HOECHST AKTIENGESELLSCHAFT (DE) 1986-03-18 US claimed
EP-0169466-A2 Mixture of xanthin derivatives and O-acetyl-salicylic acid, or their pharmacologically acceptable salts, and its use HOECHST AKTIENGESELLSCHAFT (DE) 1986-01-29 EP claimed
US-4515795-A INSUFFICIENCY OF CEREBRAL BLOOD FLOW HOECHST AKTIENGESELLSCHAFT (DE) 1985-05-07 US claimed
US-4189469-A Pharmaceutical compositions HOECHST AKTIENGESELLSCHAFT (DE) 1980-02-19 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS HDAC3, HDAC1, HDAC4 ADORA2B 1595/4885TNF 4596/4885USP2 2840/4885
US-20040013609-A1 For identification of substances for treatment or prevention of insufficient longitudinal growth of eye(hypermetropia) or excessive longitudinal growth of eye(myopia); involves measurement of effect on retinal pigment epithelium RYR1, ATP2A2, ATP2A1 ADORA2B 826/4885TNF 1783/4885USP2 2776/4885
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS HDAC1, HDAC7, HDAC5 ADORA2B 3296/4885TNF 3852/4885USP2 1827/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.