SCHEMBL6803451

SCHEMBL6803451

COC(=O)C(Cc1c[nH]c(=O)nc1NC(=O)c1c(Cl)cccc1Cl)NC(=O)N1CCC(n2c(=O)n(C)c3ccccc32)CC1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 9/20 0.40
CYP3A4 P08684 8/20 0.39
GAA P10253 1/20 0.39
HSD11B1 P28845 1/20 0.37
TNKS O95271 1/20 0.36
PARP1 P09874 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
OGFRL1 Q5TC84 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CTSS P25774 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6807473 0.93 CALCRL (0.41) CALCRLCYP3A4TNKSPARP1PARP2
SCHEMBL6803011 0.89 CALCRL (0.52) CALCRLCYP3A4HSD11B1
SCHEMBL6807774 0.87 HSD11B1 (0.41) CALCRLCYP3A4HSD11B1TNKSPARP1
SCHEMBL6807485 0.85 ITGB2 (0.41) CALCRLCYP3A4HSD11B1TNKSPARP1
SCHEMBL6807946 0.85 GAA (0.44) CYP3A4GAACYP2D6CYP2C9CYP2C19
SCHEMBL6807751 0.84 CYP3A4 (0.40) CALCRLCYP3A4GAACYP2D6CYP2C9
SCHEMBL6807625 0.84 MEN1 (0.47) CYP3A4GAACYP2D6CYP2C9CYP2C19
SCHEMBL6808040 0.84 GAA (0.40) CALCRLCYP3A4GAACYP2D6CYP2C9
SCHEMBL6808776 0.84 CYP3A4 (0.43) CALCRLCYP3A4CYP2D6
SCHEMBL6807454 0.83 GAA (0.42) CYP3A4GAACYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient TORAY INDUSTRIES, INC. (JP) 2004-02-26 US disclosed
EP-1323709-A1 UREA DERIVATIVE AND ADHESIVE-MOLECULE INHIBITOR CONTAINING THE SAME AS ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2003-07-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient ICAM1, VCAM1, EPCAM CALCRL 1811/4885CYP3A4 3783/4885GAA 2094/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.