SCHEMBL6807774

SCHEMBL6807774

COc1cccc(OC)c1C(=O)Nc1nc(=O)[nH]cc1CC(NC(=O)N1CCC(n2c(=O)n(C)c3ccccc32)CC1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.41
CALCRL Q16602 9/20 0.40
CYP3A4 P08684 3/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
TNKS O95271 1/20 0.38
PARP1 P09874 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
ECE1 P42892 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
PIK3CA P42336 1/20 0.35
POLB P06746 1/20 0.35
BRPF1 P55201 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6807485 0.92 ITGB2 (0.41) HSD11B1CALCRLCYP3A4TNKSPARP1
SCHEMBL6807459 0.91 C5AR1 (0.41) CALCRLCYP3A4DRD2DRD4DRD3
SCHEMBL6807473 0.91 CALCRL (0.41) CALCRLCYP3A4TNKSPARP1PARP2
SCHEMBL6808589 0.90 CALCRL (0.52) HSD11B1CALCRLCYP3A4DRD2DRD4
SCHEMBL6803451 0.87 CALCRL (0.40) HSD11B1CALCRLCYP3A4TNKSPARP1
SCHEMBL6807848 0.86 TACR1 (0.40) ECE1ITGB1ITGA4POLB
SCHEMBL6808312 0.86 HSD17B10 (0.42) HSD11B1TNKSPARP1ECE1ITGB1
SCHEMBL6808899 0.85 KMT2A (0.41) ECE1ITGB1ITGA4
SCHEMBL6809212 0.85 POLB (0.53) ECE1POLB
SCHEMBL6802705 0.85 KMT2A (0.42) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient TORAY INDUSTRIES, INC. (JP) 2004-02-26 US disclosed
EP-1323709-A1 UREA DERIVATIVE AND ADHESIVE-MOLECULE INHIBITOR CONTAINING THE SAME AS ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2003-07-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient ICAM1, VCAM1, EPCAM HSD11B1 3877/4885CALCRL 1811/4885CYP3A4 3783/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.