SCHEMBL6804455

SCHEMBL6804455

COc1ccc(-n2ncc(-c3nc4c(C(N)=O)cccc4[nH]3)c2C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.59
PLA2G2A P14555 1/20 0.59
ALOX15 P16050 1/20 0.59
PTGS2 P35354 1/20 0.59
CHEK2 O96017 1/20 0.46
PKN1 Q16512 1/20 0.46
PKN2 Q16513 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587344 0.88 PARP1 (0.43) PARP1PLA2G2AALOX15PTGS2
SCHEMBL6804463 0.85 FLT3 (0.42) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL6802778 0.80 PARP1 (0.61) PARP1CHEK2PKN1PKN2
SCHEMBL6807418 0.78 PARP1 (0.53) PARP1CHEK2PKN1PKN2
SCHEMBL6807472 0.77 PARP1 (0.56) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL7319077 0.76 PARP1 (1.00) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL6810588 0.76 PARP1 (0.58) PARP1CHEK2PKN1PKN2
SCHEMBL6806910 0.75 PARP1 (0.60) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL6804961 0.73 PARP1 (0.72) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL28451458 0.71 STK33 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed