SCHEMBL680578

SCHEMBL680578

Cc1cc(-c2ccccc2)c(C(=O)O)c(=O)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.49
PDE4B Q07343 1/20 0.49
PDE4C Q08493 1/20 0.49
PDE4D Q08499 1/20 0.49
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
KDM4E B2RXH2 9/20 0.45
GAA P10253 4/20 0.45
ALDH1A1 P00352 4/20 0.45
HPGD P15428 2/20 0.45
GALR3 O60755 1/20 0.45
LMNA P02545 3/20 0.45
MAPT P10636 3/20 0.45
HTT P42858 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
PRF1 P14222 1/20 0.40
GLA P06280 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PARP1 P09874 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313188 0.88 PIN1 (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL19946295 0.81 KDM4E (0.55) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL31686363 0.80 AKR1C3 (0.44) HTTMEN1KMT2A
SCHEMBL6535444 0.79 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20568185 0.77 ALDH1A1 (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL3528049 0.74 ALDH1A1 (0.61) KDM4EGAAALDH1A1HPGDLMNA
SCHEMBL19946214 0.74 MET (0.53) KDM4EGAAALDH1A1HPGDLMNA
SCHEMBL3504485 0.74 PDE3B (0.56) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7276070 0.73 PDE3B (0.61) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL6029149 0.73 TDP1 (0.43) KDM4EGAAALDH1A1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3154944-B1 SUBSTITUTED PYRIDINONES AS MGAT2 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-03-14 EP disclosed
EP-2310382-B1 AMIDOPHENOXYINDAZOLES USEFUL AS INHIBITORS OF C-MET LILLY CO ELI (US) 2012-02-22 EP disclosed