SCHEMBL680594

SCHEMBL680594

CS(=O)(=O)NC(=O)c1ccc(Oc2ccc(F)c(C(F)(F)F)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 13/20 0.52
SCN5A Q14524 3/20 0.52
PTPN1 P18031 1/20 0.47
HDAC8 Q9BY41 1/20 0.46
EPHX2 P34913 2/20 0.42
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
TAS1R2 Q8TE23 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL371116 0.86 SCN9A (0.67) SCN9ASCN5APTPN1HDAC8
SCHEMBL680206 0.85 SOS1 (0.50) SCN9APTPN1
SCHEMBL16319279 0.85 SCN9A (0.56) SCN9ASCN5A
SCHEMBL16319644 0.83 AR (0.58) SCN9ASCN5A
SCHEMBL679799 0.83 SCN9A (0.48) SCN9ASCN5APTPN1
SCHEMBL680674 0.82 SCN9A (0.57) SCN9ASCN5A
SCHEMBL680717 0.80 MAPK14 (0.56) SCN9ASCN5APTPN1
SCHEMBL703171 0.80 BCL2L1 (0.59) SCN9ASCN5APTPN1
SCHEMBL679943 0.80 SCN9A (0.57) SCN9ASCN5A
SCHEMBL678827 0.79 SCN9A (0.58) SCN9ASCN5APTPN1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010207-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 13/4885SCN5A 5/4885PTPN1 404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.