SCHEMBL16319644

SCHEMBL16319644

CS(=O)(=O)NC(=O)c1ccc(Oc2ccc(C#N)c(C(F)(F)F)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 15/20 0.58
PLA2G7 Q13093 1/20 0.49
SCN9A Q15858 3/20 0.48
SCN5A Q14524 1/20 0.48
FPR2 P25090 1/20 0.48
ESRRA P11474 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319948 0.86 SCN9A (0.51) ARSCN9ASCN5A
SCHEMBL680594 0.83 SCN9A (0.52) SCN9ASCN5A
SCHEMBL371116 0.82 SCN9A (0.67) SCN9ASCN5A
SCHEMBL680332 0.82 SCN9A (0.53) ARSCN9ASCN5A
SCHEMBL16319655 0.82 PLA2G7 (0.62) ARPLA2G7SCN9ASCN5A
SCHEMBL4174817 0.82 AR (0.68) ARESRRA
SCHEMBL365304 0.80 SCN9A (0.46) ARSCN9ASCN5A
SCHEMBL680479 0.77 SCN9A (0.50) ARPLA2G7SCN9ASCN5A
SCHEMBL680717 0.76 MAPK14 (0.56) ARSCN9ASCN5A
SCHEMBL679345 0.75 SCN9A (0.51) PLA2G7SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed