SCHEMBL6806004

SCHEMBL6806004

NC(=O)c1cccc2nc(-c3cnccc3OCCN3CCNCC3)[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.40
DHODH Q02127 1/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
TBXAS1 P24557 1/20 0.38
HTR1A P08908 1/20 0.37
DRD2 P14416 3/20 0.37
DRD3 P35462 3/20 0.37
PDE5A O76074 2/20 0.37
TBK1 Q9UHD2 1/20 0.37
ROCK1 Q13464 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
MELK Q14680 1/20 0.36
CHEK2 O96017 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6799974 0.96 PARP1 (0.41) PARP1DHODHKDM4EALDH1A1TDP1
SCHEMBL6806306 0.93 PARP1 (0.47) PARP1DHODHKDM4ETBXAS1HTR1A
SCHEMBL6810662 0.92 PARP1 (0.49) PARP1DHODHKDM4ETBXAS1HTR1A
SCHEMBL6810121 0.91 HTR1A (0.41) PARP1DHODHKDM4EALDH1A1TBXAS1
SCHEMBL6809941 0.88 PARP1 (0.48) PARP1DHODHKDM4EALDH1A1HTR1A
SCHEMBL6802868 0.88 HTR1A (0.45) PARP1DHODHKDM4EALDH1A1TDP1
SCHEMBL6805803 0.88 PARP1 (0.49) PARP1DHODHKDM4EALDH1A1HTR1A
SCHEMBL6806267 0.87 HTR1A (0.43) PARP1KDM4EALDH1A1HTR1ADRD2
SCHEMBL6806003 0.87 PARP1 (0.56) PARP1DHODHROCK1CHEK2
SCHEMBL6806140 0.84 DRD2 (0.44) PARP1KDM4EALDH1A1TDP1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed