SCHEMBL6806441

SCHEMBL6806441

NC(=O)c1cccc2nc(-c3ccc(N4CCCN(Cc5ccccc5)CC4)nc3)[nH]c12

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.70
AURKA O14965 2/20 0.70
KDR P35968 2/20 0.70
PARP1 P09874 9/20 0.49
OPRM1 P35372 1/20 0.49
OPRK1 P41145 1/20 0.49
DHODH Q02127 1/20 0.46
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
DGAT1 O75907 1/20 0.42
KCNH2 Q12809 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
NPBWR1 P48145 1/20 0.41
MCHR1 Q99705 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
BCHE P06276 1/20 0.41
CHEK2 O96017 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805222 0.97 AURKA (0.75) AURKBAURKAKDRPARP1OPRM1
SCHEMBL6806887 0.89 AURKA (0.60) AURKBAURKAKDRPARP1OPRM1
SCHEMBL6802572 0.88 AURKA (0.64) AURKBAURKAKDRPARP1OPRM1
SCHEMBL3585487 0.88 PARP1 (0.54) AURKBAURKAKDRPARP1DHODH
SCHEMBL6810130 0.88 AURKA (0.54) AURKBAURKAKDRPARP1NPC1
SCHEMBL6804570 0.86 AURKA (0.72) AURKBAURKAKDRPARP1OPRM1
SCHEMBL6806434 0.86 AURKB (0.93) AURKBAURKAKDRPARP1DHODH
SCHEMBL6805914 0.86 AURKA (0.55) AURKBAURKAKDRPARP1DHODH
SCHEMBL6809975 0.85 AURKA (0.54) AURKBAURKAKDRPARP1DHODH
SCHEMBL6806391 0.85 AURKA (0.54) AURKBAURKAKDRPARP1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed