SCHEMBL680695

SCHEMBL680695

Cc1cc(-c2cc3c(cnn3C)cc2Oc2ccc(N)cc2F)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 2/20 0.41
PLK4 O00444 1/20 0.41
NTRK1 P04629 1/20 0.41
RET P07949 1/20 0.41
MET P08581 1/20 0.41
KDR P35968 1/20 0.41
FLT3 P36888 1/20 0.41
MST1R Q04912 1/20 0.41
DDR1 Q08345 1/20 0.41
MERTK Q12866 1/20 0.41
CAMK4 Q16566 1/20 0.41
DDR2 Q16832 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
AAK1 Q2M2I8 1/20 0.37
GRM2 Q14416 2/20 0.35
ALOX5AP P20292 3/20 0.35
FEN1 P39748 3/20 0.35
TRPA1 O75762 1/20 0.34
PDE10A Q9Y233 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL680085 0.84 S1PR4 (0.44) AXLPLK4NTRK1RETMET
SCHEMBL680022 0.83 CYP11B1 (0.43) AXLPLK4NTRK1RETMET
SCHEMBL23081429 0.82 AXL (0.41) AXLPLK4NTRK1RETMET
SCHEMBL680039 0.82 PLK4 (0.55) AXLPLK4NTRK1RETMET
SCHEMBL680260 0.79 TLR8 (0.46) AAK1ALOX5APFEN1TRPA1
SCHEMBL680999 0.78 PLK4 (0.42) AXLPLK4NTRK1RETMET
SCHEMBL30896357 0.77 CDC7 (0.41) GRM2TRPA1ARIRAK4USP7
SCHEMBL31613173 0.74 CDC7 (0.41) GRM2TRPA1ARIRAK4USP7
SCHEMBL680838 0.74 SCN9A (0.45) AXLPLK4NTRK1RETMET
SCHEMBL680681 0.74 CACNA1H (0.42) AXLPLK4NTRK1RETMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2310382-B1 AMIDOPHENOXYINDAZOLES USEFUL AS INHIBITORS OF C-MET LILLY CO ELI (US) 2012-02-22 EP disclosed