SCHEMBL6807066

SCHEMBL6807066

O=Cc1ccc(C(F)(F)F)cc1C1CCCC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.49
CHRNB2 P17787 2/20 0.41
CHRNA4 P43681 2/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
PNMT P11086 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
CSNK1D P48730 1/20 0.38
HTR2A P28223 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TSHR P16473 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27486622 0.93 CHRNB2 (0.44) PTGDR2CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL19974321 0.86 HTR2C (0.51) CHRNB2CHRNA4CHRNB4CHRNA3PNMT
SCHEMBL19974334 0.81 RBP4 (0.45) PTGDR2HTR2AMRGPRX4
SCHEMBL20303392 0.80 CHRNB2 (0.44) PTGDR2CHRNB2CHRNA4CHRNB4CHRNA3
Trifluoroacetic Acid SCHEMBL21271258 0.80 HTR2C (0.44) PTGDR2CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL28897105 0.78 CA1 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3PNMT
SCHEMBL19974343 0.78 PTGDR2 (0.45) PTGDR2KMT2AMRGPRX4
SCHEMBL27848652 0.76 PTGDR2 (0.43) PTGDR2CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL20503456 0.76 CHRNB2 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3PNMT
SCHEMBL29170876 0.75 KMT2A (0.40) PNMTNOS3NOS1NOS2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470102-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) Applied Research Systems ARS Holding N.V. (AN) 2004-10-27 EP disclosed
WO-2003064376-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2003-08-07 WO disclosed