SCHEMBL6807459

SCHEMBL6807459

COc1cccc(OC)c1C(=O)Nc1nc(=O)[nH]cc1CC(NC(=O)N1CCC(n2c(=O)n(Cc3ccccc3)c3ccccc32)CC1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 6/20 0.41
CYP3A4 P08684 7/20 0.41
CYP2D6 P10635 5/20 0.41
CALCRL Q16602 4/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
POLB P06746 1/20 0.36
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6808858 0.92 C5AR1 (0.46) C5AR1CYP3A4CYP2D6CALCRLOPRM1
SCHEMBL6807774 0.91 HSD11B1 (0.41) CYP3A4CALCRLDRD2DRD4DRD3
SCHEMBL6808776 0.91 CYP3A4 (0.43) C5AR1CYP3A4CYP2D6CALCRLPOLB
SCHEMBL6808589 0.87 CALCRL (0.52) CYP3A4CALCRLDRD2DRD4DRD3
SCHEMBL6809212 0.85 POLB (0.53) POLB
SCHEMBL6807848 0.85 TACR1 (0.40) POLBITGB1ITGA4
SCHEMBL6807473 0.84 CALCRL (0.41) CYP3A4CALCRLPOLBITGB1ITGA4
SCHEMBL6807485 0.83 ITGB2 (0.41) CYP3A4CALCRLPOLB
SCHEMBL6808312 0.83 HSD17B10 (0.42) POLBITGB1ITGA4
SCHEMBL6808899 0.82 KMT2A (0.41) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient TORAY INDUSTRIES, INC. (JP) 2004-02-26 US disclosed
EP-1323709-A1 UREA DERIVATIVE AND ADHESIVE-MOLECULE INHIBITOR CONTAINING THE SAME AS ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2003-07-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient ICAM1, VCAM1, EPCAM C5AR1 930/4885CYP3A4 3783/4885CYP2D6 4452/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.