SCHEMBL680979

SCHEMBL680979

CCOC(=O)c1ccc(C)n(-c2ccc(F)cc2)c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.56
HTT P42858 2/20 0.56
LMNA P02545 3/20 0.49
RAB9A P51151 3/20 0.49
NPC1 O15118 2/20 0.49
POLB P06746 1/20 0.49
CHRNA7 P36544 2/20 0.48
MAPK1 P28482 1/20 0.48
KDM4E B2RXH2 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ALDH1A1 P00352 3/20 0.46
TP53 P04637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MAPT P10636 4/20 0.45
GABRA2 P47869 1/20 0.45
GABRB2 P47870 1/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
APP P05067 1/20 0.45
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23629459 0.86 CHRNA7 (0.52) HPGDHTTLMNARAB9ANPC1
SCHEMBL23629499 0.86 KDM4E (0.50) HPGDHTTLMNARAB9ANPC1
SCHEMBL5762071 0.86 MAPK1 (0.65) HPGDHTTLMNARAB9ANPC1
SCHEMBL3061680 0.86 ALDH1A1 (0.57) HPGDHTTRAB9AMAPK1KDM4E
SCHEMBL23629430 0.84 POLB (0.45) HPGDHTTLMNARAB9ANPC1
SCHEMBL6212346 0.82 MAPK1 (0.60) HPGDHTTRAB9ANPC1CHRNA7
SCHEMBL679510 0.81 NOTUM (0.60) HPGDLMNAPOLBKDM4EL3MBTL1
SCHEMBL23146843 0.80 POLB (0.52) HPGDLMNARAB9ANPC1POLB
SCHEMBL16092699 0.80 POLB (0.49) HPGDHTTLMNARAB9ANPC1
SCHEMBL14969108 0.80 ALDH1A1 (0.51) HPGDHTTLMNARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113195471-B Polysubstituted pyridone derivative and application thereof in medicine 苏州浦合医药科技有限公司 2023-05-02 CN disclosed
CN-110627796-B Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2022-07-12 CN disclosed
US-20210355107-A1 MULTI-SUBSTITUTED PYRIDONE DERIVATIVES AND MEDICAL USE THEREOF BEIJING YUEZHIKANGTAI BIOMEDICINES CO LTD (CN) 2021-11-18 US disclosed
US-20210355107-A1 MULTI-SUBSTITUTED PYRIDONE DERIVATIVES AND MEDICAL USE THEREOF BEIJING YUEZHIKANGTAI BIOMEDICINES CO LTD (CN) 2021-11-18 US disclosed
CN-113195471-A Polysubstituted pyridone derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2021-07-30 CN disclosed
EP-3845527-A1 MULTI-SUBSTITUTED PYRIDONE DERIVATIVES AND MEDICAL USE THEREOF Beijing Yuezhikangtai Biomedicines Co., Ltd. (CN) 2021-07-07 EP disclosed
EP-3845527-A1 MULTI-SUBSTITUTED PYRIDONE DERIVATIVES AND MEDICAL USE THEREOF Beijing Yuezhikangtai Biomedicines Co., Ltd. (CN) 2021-07-07 EP disclosed
WO-2020042618-A1 MULTI-SUBSTITUTED PYRIDONE DERIVATIVES AND MEDICAL USE THEREOF 北京越之康泰生物医药科技有限公司 2020-03-05 WO disclosed
WO-2020042618-A1 MULTI-SUBSTITUTED PYRIDONE DERIVATIVES AND MEDICAL USE THEREOF 北京越之康泰生物医药科技有限公司 2020-03-05 WO disclosed
CN-110627796-A Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2019-12-31 CN disclosed
US-RE43878-E1 Amidophenoxyindazoles useful as inhibitors of c-Met ELI LILLY AND COMPANY (US) 2012-12-25 US disclosed
EP-2310382-B1 AMIDOPHENOXYINDAZOLES USEFUL AS INHIBITORS OF C-MET LILLY CO ELI (US) 2012-02-22 EP disclosed
US-8030302-B2 Amidophenoxyindazoles useful as inhibitors of c-Met ELI LILLY AND COMPANY (US) 2011-10-04 US disclosed
US-20100022529-A1 AMIDOPHENOXYINDAZOLES USEFUL AS INHIBITORS OF C-MET ELI LILLY AND COMPANY 2010-01-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210355107-A1 MULTI-SUBSTITUTED PYRIDONE DERIVATIVES AND MEDICAL USE THEREOF PDXK, ITK, JAK1 HPGD 577/4885HTT 3897/4885LMNA 3969/4885
US-20100022529-A1 AMIDOPHENOXYINDAZOLES USEFUL AS INHIBITORS OF C-MET MET, MYCBP, MYC HPGD 3623/4885HTT 4635/4885LMNA 4448/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.