SCHEMBL681350

SCHEMBL681350

C=C(C(C)C)[C@H](CN1C[C@@H](C)N[C@@H](C)C1)c1ccc(Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
THRB P10828 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MDM2 Q00987 1/20 0.36
SLC6A9 P48067 3/20 0.35
NTSR1 P30989 1/20 0.35
MLNR O43193 4/20 0.35
CYP3A4 P08684 2/20 0.35
SIGMAR1 Q99720 2/20 0.34
POLB P06746 1/20 0.34
HSD11B1 P28845 1/20 0.33
S1PR1 P21453 1/20 0.33
OPRD1 P41143 1/20 0.33
TACR1 P25103 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL680169 1.00 MEN1 (0.38) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL680790 0.87 MEN1 (0.38) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL681295 0.87 MEN1 (0.38) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL681616 0.85 ALDH1A1 (0.54) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL680168 0.85 ALDH1A1 (0.54) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL12188597 0.84 BRD4 (0.40) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL683331 0.84 BRD4 (0.40) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL681313 0.84 MEN1 (0.37) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL681578 0.84 MEN1 (0.37) MEN1ALDH1A1THRBKMT2ASMN1; SMN2
SCHEMBL2738604 0.83 MEN1 (0.39) MEN1ALDH1A1THRBKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9359340-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as Akt protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2016-06-07 US disclosed
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed