SCHEMBL681584

SCHEMBL681584

C=C(C(C)C)[C@H](CNC(C)C)c1ccc(C(F)(F)F)cc1F

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 14/20 0.50
ADRB2 P07550 2/20 0.39
ADRB1 P08588 2/20 0.39
ADRB3 P13945 2/20 0.39
GPR139 Q6DWJ6 2/20 0.37
SLC6A4 P31645 1/20 0.35
TRPV1 Q8NER1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681232 0.87 PDE2A (0.50) PDE2AADRB2ADRB1ADRB3GPR139
SCHEMBL12188384 0.86 PDE2A (0.51) PDE2AADRB2ADRB1ADRB3GPR139
SCHEMBL2738439 0.85 PDE2A (0.50) PDE2AADRB2ADRB1ADRB3GPR139
SCHEMBL681790 0.83 PDE2A (0.54) PDE2AGPR139SLC6A4
SCHEMBL17803802 0.83 ADRB2 (0.41) ADRB2ADRB1ADRB3GPR139
SCHEMBL681254 0.82 PDE2A (0.45) PDE2ASLC6A4
SCHEMBL681752 0.82 ADRB2 (0.40) ADRB2ADRB1ADRB3
SCHEMBL681362 0.82 ADRB2 (0.40) ADRB2ADRB1ADRB3
SCHEMBL681744 0.82 ADRB2 (0.40) ADRB2ADRB1ADRB3
SCHEMBL681594 0.80 CA1 (0.38) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed