SCHEMBL681790

SCHEMBL681790

C=C(C(C)C)[C@H](CN)c1ccc(C(F)(F)F)cc1F

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 14/20 0.54
IDO1 P14902 2/20 0.39
SLC6A4 P31645 1/20 0.37
GPR139 Q6DWJ6 1/20 0.36
PNMT P11086 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681320 0.86 PDE2A (0.54) PDE2AIDO1SLC6A4GPR139PNMT
SCHEMBL12188449 0.83 PDE2A (0.54) PDE2AIDO1GPR139PNMT
SCHEMBL681584 0.83 PDE2A (0.50) PDE2ASLC6A4GPR139
SCHEMBL681205 0.82 PDE2A (0.49) PDE2ASLC6A4
SCHEMBL2738655 0.81 PDE2A (0.51) PDE2AIDO1GPR139PNMT
SCHEMBL17803817 0.81 ADRA1A (0.35) GPR139
SCHEMBL681363 0.80 KCNH2 (0.38)
SCHEMBL680198 0.80 APLNR (0.44)
SCHEMBL681254 0.78 PDE2A (0.45) PDE2ASLC6A4
SCHEMBL18636315 0.77 PDE2A (0.60) PDE2AIDO1PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed