SCHEMBL6817879

SCHEMBL6817879

CCCCCNc1nc(Cl)nc2c1ncn2C1CCCC1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.70
ADORA3 P0DMS8 4/20 0.50
ADORA1 P30542 3/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
YTHDC1 Q96MU7 2/20 0.48
CDK1 P06493 2/20 0.47
TDP1 Q9NUW8 1/20 0.46
FLT3 P36888 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8110131 0.99 CTSL (0.72) CTSLADORA3ADORA1HDAC1HDAC2
SCHEMBL6820572 0.99 CTSL (0.72) CTSLADORA3ADORA1HDAC1HDAC2
SCHEMBL8204168 0.99 CTSL (0.72) CTSLADORA3ADORA1HDAC1HDAC2
SCHEMBL6817663 0.99 CTSL (0.72) CTSLADORA3ADORA1HDAC1HDAC2
SCHEMBL6947217 0.99 CTSL (0.72) CTSLADORA3ADORA1HDAC1HDAC2
SCHEMBL6820593 0.97 CTSL (0.66) CTSLADORA3ADORA1HDAC1HDAC2
SCHEMBL6817775 0.92 CTSL (0.59) CTSLADORA3ADORA1YTHDC1CDK1
SCHEMBL6824196 0.89 CTSL (0.56) CTSLADORA3ADORA1YTHDC1CDK1
SCHEMBL6945264 0.88 CTSL (0.56) CTSLADORA3ADORA1YTHDC1CDK1
SCHEMBL6949990 0.88 CTSL (0.56) CTSLADORA3ADORA1YTHDC1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056745-B1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMA INC (US) 2004-06-16 EP disclosed
US-6413974-B1 INHIBITORS OF CYCLIN DEPENDENT KINASES, PARTICULARLY CDK-2; PREVENTING APOPTOSIS IN NEURONAL CELLS; ANTINEOPLASTIC AGENTS; NEURONAL INJURY AND DEGENERATION; CEREBROVASCULAR DISEASE AVENTIS PHARMACEUTICALS INC. 2002-07-02 US disclosed
EP-1056745-A2 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES Aventis Pharmaceuticals Inc. (US) 2000-12-06 EP disclosed
WO-1999043676-A2 6,9-DISUBSTITUTED 2-[TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMACEUTICALS INC. (US) 1999-09-02 WO disclosed