SCHEMBL6818399

SCHEMBL6818399

COc1ccccc1-c1cc2c(C(=O)Nc3ccc(C#N)cc3C(=O)O)noc2cc1C(C)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 5/20 0.46
TSHR P16473 3/20 0.39
MEN1 O00255 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 3/20 0.39
TP53 P04637 2/20 0.39
HTT P42858 1/20 0.39
LRRK2 Q5S007 1/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ALB P02768 1/20 0.37
MAPT P10636 2/20 0.37
DHODH Q02127 1/20 0.37
KDM4E B2RXH2 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
GPR35 Q9HC97 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822443 0.90 HIF1A (0.46) HIF1ATSHRMEN1ALDH1A1KMT2A
SCHEMBL6818998 0.89 HIF1A (0.39) HIF1AALDH1A1HTTLRRK2HPGD
SCHEMBL6818846 0.89 ALDH1A1 (0.39) HIF1AALDH1A1TP53HTTLRRK2
SCHEMBL6813822 0.88 AGPAT2 (0.37) HIF1AMEN1KMT2ATP53HTT
SCHEMBL6822476 0.88 HIF1A (0.44) HIF1ATSHRMEN1ALDH1A1KMT2A
SCHEMBL6817520 0.87 HIF1A (0.43) HIF1ATSHRMEN1ALDH1A1KMT2A
SCHEMBL6818178 0.87 HIF1A (0.43) HIF1ATSHRMEN1ALDH1A1KMT2A
SCHEMBL6817683 0.86 HIF1A (0.44) HIF1ATSHRMEN1ALDH1A1KMT2A
SCHEMBL6818353 0.86 DHODH (0.37) HIF1ATSHRMEN1KMT2ATP53
SCHEMBL6818297 0.86 HIF1A (0.45) HIF1ATSHRMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018428-A1 ANTIBACTERIAL BENZOIC ACID DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO disclosed