SCHEMBL6818521

SCHEMBL6818521

COCCCCNc1nccc(-c2ccc(OC)cc2C)c1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.44
NPC1 O15118 1/20 0.38
LMNA P02545 3/20 0.37
ALDH1A1 P00352 3/20 0.36
HTT P42858 1/20 0.36
HTR1A P08908 2/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
EGLN1 Q9GZT9 1/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
RAD52 P43351 1/20 0.35
RECQL P46063 1/20 0.35
BLM P54132 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6817779 0.89 MAPT (0.43) MAPTNPC1LMNAALDH1A1HTT
SCHEMBL6817636 0.85 BRD4 (0.37) MAPTNPC1LMNAALDH1A1KDM5A
SCHEMBL6817889 0.84 MAPT (0.40) MAPTNPC1LMNAALDH1A1HTT
SCHEMBL6818841 0.84 MAPT (0.40) MAPTLMNAALDH1A1HTTEGLN1
SCHEMBL6819213 0.82 MEN1 (0.39) MAPTNPC1LMNAALDH1A1HTT
SCHEMBL6083484 0.82 CRHR1 (0.38) MAPTNPC1ALDH1A1HTTKDM5A
SCHEMBL6082375 0.81 CRHR1 (0.44) MAPTTDP1KDM4E
SCHEMBL6817723 0.79 CRHR1 (0.38) MAPTNPC1LMNAALDH1A1HTT
SCHEMBL6818033 0.78 MAPT (0.43) MAPTNPC1LMNAALDH1A1HTT
SCHEMBL6818822 0.78 MAPT (0.39) MAPTLMNAALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed