SCHEMBL6818666

SCHEMBL6818666

Cc1cc(Cc2ccc(C(=O)O)cc2)c(=O)n2c1CC(C(=O)NCc1ccccc1)=C2.Cc1cc(Cc2ccc(C(=O)O)cc2)c(=O)n2cc(C(=O)NCc3ccccc3)sc12

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 10/20 0.44
NR1H4 Q96RI1 1/20 0.36
LMNA P02545 2/20 0.36
RXFP1 Q9HBX9 2/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
HTT P42858 1/20 0.35
MAPK10 P53779 1/20 0.35
CASP7 P55210 1/20 0.35
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35
PHGDH O43175 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6818671 0.93 TRPA1 (0.42) TRPA1LMNARXFP1POLBMAPT
SCHEMBL6488185 0.89 TRPA1 (0.53) TRPA1NR1H4LMNARXFP1POLB
SCHEMBL6486746 0.89 NR1H4 (0.45) NR1H4LMNAPOLBMAPTALDH1A1
SCHEMBL6476120 0.77 TRPA1 (0.54) TRPA1LMNARXFP1POLBMAPT
SCHEMBL6483921 0.73 MAPT (0.45) NR1H4LMNARXFP1POLBMAPT
SCHEMBL6814150 0.72 TRPA1 (0.51) TRPA1MAPT
SCHEMBL6483805 0.72 KLK1 (0.47) NR1H4RXFP1MAPTALDH1A1HPGD
SCHEMBL6488181 0.71 NR1H4 (0.44) NR1H4LMNAMAPTALDH1A1HPGD
SCHEMBL6817760 0.71 MAPT (0.38) NR1H4LMNARXFP1POLBMAPT
SCHEMBL6487093 0.71 NR1H4 (0.46) NR1H4POLBALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014908-A1 HETEROBICYLCIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed