SCHEMBL6820248

SCHEMBL6820248

Cc1c(OCCN(C)C)c2cc(Cl)ccc2n1C(=O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.47
PTGS1 P23219 4/20 0.47
ABCB1 P08183 2/20 0.47
KDM4E B2RXH2 2/20 0.46
PPARG P37231 4/20 0.44
AKR1C3 P42330 3/20 0.44
AKR1C2 P52895 3/20 0.44
LMNA P02545 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
HIF1A Q16665 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PTGES O14684 1/20 0.44
ABCC3 O15438 1/20 0.44
ABCC4 O15439 1/20 0.44
ABCB11 O95342 1/20 0.44
MT-CO2 P00403 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6820242 0.93 KDM4E (0.45) PTGS2PTGS1ABCB1KDM4ETDP1
SCHEMBL6919614 0.89 PTGS2 (0.46) PTGS2ABCB1KDM4EMEN1KMT2A
SCHEMBL6821172 0.88 ELANE (0.45) KDM4ELMNACYP1A2CYP2D6CYP2C9
SCHEMBL6817370 0.88 P2RX4 (0.46) PTGS2PTGS1ABCB1LMNACYP1A2
SCHEMBL6817298 0.87 LMNA (0.61) PTGS2PTGS1ABCB1KDM4EPPARG
SCHEMBL6820214 0.85 MEN1 (0.41) PTGS2KDM4EPPARGMEN1KMT2A
SCHEMBL3553237 0.85 KDM4E (0.44) KDM4ECYP1A2MEN1KMT2ATDP1
SCHEMBL6820272 0.84 KDM4E (0.46) ABCB1KDM4EMEN1KMT2ATDP1
SCHEMBL6821012 0.82 KDM4E (0.41) ABCB1KDM4ELMNACYP1A2CYP2D6
SCHEMBL6821037 0.80 ABCB1 (0.43) PTGS2ABCB1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048331-A1 N-ARYLALKYL-3-AMINOALKOXYINDOLES AND THEIR USE AS 5-HT LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2004-06-10 WO disclosed