SCHEMBL6820586

SCHEMBL6820586

Clc1nc(NCC2CCCCO2)c2ncn(C3CCCC3)c2n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 1/20 0.57
ADORA3 P0DMS8 5/20 0.48
ADORA2A P29274 5/20 0.48
ADORA1 P30542 5/20 0.48
CDK1 P06493 3/20 0.47
CCNB2 O95067 1/20 0.47
CCNE2 O96020 1/20 0.47
CDK4 P11802 1/20 0.47
CCNB1 P14635 1/20 0.47
CCND1 P24385 1/20 0.47
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47
CCNB3 Q8WWL7 1/20 0.47
CTSL P07711 3/20 0.46
NT5E P21589 1/20 0.44
ADORA2B P29275 4/20 0.44
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
MAPK1 P28482 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18587836 0.87 YTHDC1 (0.66) YTHDC1ADORA3ADORA2AADORA1MEN1
SCHEMBL29664966 0.87 YTHDC1 (0.66) YTHDC1ADORA3ADORA2AADORA1MEN1
SCHEMBL6821032 0.84 ADORA3 (0.64) YTHDC1ADORA3ADORA2AADORA1CDK1
SCHEMBL6817815 0.83 ADORA3 (0.60) YTHDC1ADORA3ADORA2AADORA1CDK1
SCHEMBL17902904 0.80 YTHDC1 (0.72) YTHDC1ADORA3ADORA2AADORA1CDK1
SCHEMBL6818080 0.80 ADORA3 (0.61) YTHDC1ADORA3ADORA2AADORA1CDK1
Hydrochloric Acid SCHEMBL6817867 0.80 CDK2 (0.75) CDK1CCNB2CCNE2CDK4CCNB1
Hydrochloric Acid SCHEMBL6817861 0.80 CDK2 (0.75) CDK1CCNB2CCNE2CDK4CCNB1
SCHEMBL6945547 0.79 ADORA3 (0.61) ADORA3ADORA2AADORA1CDK1CCNB2
SCHEMBL6817775 0.78 CTSL (0.59) YTHDC1ADORA3ADORA2AADORA1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056745-B1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMA INC (US) 2004-06-16 EP disclosed
US-6413974-B1 INHIBITORS OF CYCLIN DEPENDENT KINASES, PARTICULARLY CDK-2; PREVENTING APOPTOSIS IN NEURONAL CELLS; ANTINEOPLASTIC AGENTS; NEURONAL INJURY AND DEGENERATION; CEREBROVASCULAR DISEASE AVENTIS PHARMACEUTICALS INC. 2002-07-02 US disclosed
EP-1056745-A2 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES Aventis Pharmaceuticals Inc. (US) 2000-12-06 EP disclosed
WO-1999043676-A2 6,9-DISUBSTITUTED 2-[TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMACEUTICALS INC. (US) 1999-09-02 WO disclosed