SCHEMBL6821940

SCHEMBL6821940

Cc1c(COC(=O)c2ccccc2OS(=O)(=O)O)ccc2nc(N)nc(N)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCPS Q96C86 5/20 0.40
DHFR P00374 3/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ESR1 P03372 1/20 0.40
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
CHRM1 P11229 1/20 0.40
HPGD P15428 1/20 0.40
MAOA P21397 1/20 0.40
DRD1 P21728 1/20 0.40
ACHE P22303 1/20 0.40
PTGS1 P23219 1/20 0.40
SLC6A2 P23975 1/20 0.40
PDE4A P27815 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
BLM P54132 1/20 0.40
SLC6A3 Q01959 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6825657 0.86 DHFR (0.41) DCPSDHFRMAPTMEN1ALDH1A1
SCHEMBL6827408 0.84 KDM4E (0.44) DCPSDHFRMAPTMEN1ALDH1A1
SCHEMBL6825666 0.83 MAPT (0.41) DCPSDHFRMAPTMEN1ALDH1A1
SCHEMBL6827464 0.83 MAPT (0.46) DHFRMAPTMEN1ALDH1A1ESR1
SCHEMBL6825056 0.78 KDM4E (0.40) ALDH1A1
SCHEMBL6827375 0.78 DHFR (0.47) DHFRMAPT
SCHEMBL6827525 0.72 PTGS1 (0.45) DHFRMAPTMEN1ALDH1A1ESR1
SCHEMBL27816716 0.70 TSHR (0.62) MAPTMEN1ALDH1A1HPGDKMT2A
Benzene SCHEMBL10481612 0.68 DHFR (0.50) DCPSDHFRMAPTMEN1ALDH1A1
SCHEMBL16695948 0.68 DHFR (0.52) DHFRMAPTMEN1ALDH1A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO claimed
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO disclosed