SCHEMBL6827375

SCHEMBL6827375

Nc1nc(N)c2cc(COC(=O)c3ccccc3OS(=O)(=O)O)ccc2n1

nearest known ligand 0.66

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.47
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821942 0.84 DHFR (0.48) DHFRMAPT
SCHEMBL6827422 0.84 KDM4E (0.48) DHFRMAPT
SCHEMBL6827444 0.84 TDP1 (0.49) DHFRMAPT
SCHEMBL6748619 0.83 DHFR (0.52) DHFR
SCHEMBL6827626 0.83 TDP1 (0.56) DHFRMAPT
SCHEMBL6747477 0.82 DHFR (0.51) DHFR
SCHEMBL6750825 0.80 DHFR (0.49) DHFR
SCHEMBL6744730 0.79 DHFR (0.50) DHFR
SCHEMBL6821940 0.78 DCPS (0.40) DHFRMAPT
SCHEMBL6747511 0.76 DHFR (0.64) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO claimed
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO disclosed