SCHEMBL6825657

SCHEMBL6825657

CC(=O)Oc1ccccc1C(=O)OCc1ccc2nc(N)nc(N)c2c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.41
ALDH1A1 P00352 2/20 0.41
ESR1 P03372 2/20 0.41
HPGD P15428 2/20 0.41
PTGS1 P23219 2/20 0.41
BLM P54132 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
MEN1 O00255 1/20 0.41
CHRM2 P08172 1/20 0.41
HTR1A P08908 1/20 0.41
MAPT P10636 1/20 0.41
CHRM1 P11229 1/20 0.41
MAOA P21397 1/20 0.41
DRD1 P21728 1/20 0.41
ACHE P22303 1/20 0.41
SLC6A2 P23975 1/20 0.41
PDE4A P27815 1/20 0.41
OPRM1 P35372 1/20 0.41
DRD3 P35462 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6827408 0.98 KDM4E (0.44) DHFRALDH1A1ESR1HPGDPTGS1
SCHEMBL6825666 0.89 MAPT (0.41) DHFRALDH1A1ESR1HPGDPTGS1
SCHEMBL6821940 0.86 DCPS (0.40) DHFRALDH1A1ESR1HPGDPTGS1
SCHEMBL6827464 0.85 MAPT (0.46) DHFRALDH1A1ESR1HPGDPTGS1
SCHEMBL6825659 0.78 KDM4E (0.45) ALDH1A1ESR1HPGDPTGS1BLM
SCHEMBL6821942 0.78 DHFR (0.48) DHFRMAPTKDM4EHSD17B10LMNA
SCHEMBL6827422 0.78 KDM4E (0.48) DHFRMAPTKDM4EHSD17B10LMNA
SCHEMBL6825161 0.77 KDM4E (0.49) ALDH1A1ESR1HPGDPTGS1BLM
SCHEMBL11318544 0.70 PTGS2 (0.52) ALDH1A1ESR1HPGDPTGS1BLM
SCHEMBL11315493 0.70 KDM4E (0.54) ALDH1A1ESR1HPGDPTGS1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO claimed
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO disclosed