SCHEMBL6822445

SCHEMBL6822445

CN1C(=O)N(Cc2ccc(F)c(F)c2)Cc2nc(C(=O)O)[nH]c21.NCc1ccncc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NCOA1 Q15788 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPK1 P28482 2/20 0.35
BRD4 O60885 1/20 0.33
CYP3A4 P08684 1/20 0.33
ABCC1 P33527 1/20 0.33
CLPP Q16740 3/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
POLB P06746 2/20 0.32
DAO P14920 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
MAPK3 P27361 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6703428 0.91 ALDH1A1 (0.39) ALDH1A1KDM4EMEN1KMT2ANCOA1
SCHEMBL6822444 0.84 NAMPT (0.40) ALDH1A1KDM4EMEN1KMT2ANCOA1
Picolamine SCHEMBL6818745 0.81 S1PR3 (0.40) ALDH1A1KDM4EMEN1KMT2ATSHR
SCHEMBL6700327 0.78 CLPP (0.43) ALDH1A1CLPPPOLB
SCHEMBL6700576 0.71 CLPP (0.39) MAPK1CLPPTLR7PARP1PARP2
SCHEMBL6699940 0.70 MAPK1 (0.34) ALDH1A1MAPK1BRD4CLPPPOLB
SCHEMBL6700986 0.70 MAPK1 (0.36) ALDH1A1TSHRL3MBTL1MAPK1BRD4
SCHEMBL6699350 0.68 P2RX7 (0.35) MAPK1CYP3A4
SCHEMBL6697984 0.65 ALDH1A1 (0.36) ALDH1A1TSHRL3MBTL1MAPK1
SCHEMBL6813649 0.64 KDM5A (0.36) ALDH1A1KDM4EMEN1KMT2ANCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed